Ola kinoHoomakaukau

"Enalapril": kuhi no ka hoʻohana a me ka manaʻo. Analogs "Enalapril"

Inā 'oe i pilikia a me ke koko,, he nui loaa mai kauka koi, e lawe i ka lāʻau "enalapril" (papa). Mai mea kōkua pakele o keia lapaʻau? Mai ka waiwai o ka maʻi ( 'o ia hoʻi,' ana mai kiʻekiʻe ke koko,), a me ka mea, ua hana ma luna o kekahi mau fronts, hoihoi i ka maʻamau hana o ka mea'ōnaehana mānowai koko'ōnaehana, e kauoha ana i ke koko, hoike i ka maʻamau? E maopopo pehea papa e "Enalapril" puʻe pono no ka ike me ka oihana alakaʻi ma luna o ka hana o keia ka lapaʻauʻia. Eia hou kekahi, he helu o analogs o keia k ma kaʻeleu 'Oponopono mākou noonoo a mai ka hopena.

Description o ka la hoomalolo, i ke kalaʻana aku palapala, o ka oi aku pūnaewele a me ka dispensing ana o nā keʻena kūʻai lāʻau lapaʻau

Akala "Enalapril" puʻe hua mai ma na mea he nui mea lāʻau lapaʻau poʻe a puni ka honua. I ka papa kuhikuhiEʻeleu 'Oponopono o keia ka lapaʻauʻia ka enalapril maleate, a ma kona hui affiliation pili i ka ACE-blockers. Currently, eia nā papa me kaʻeleu 'Oponopono maʻiʻo o ka 5, 10 a me 20 mg. Aie i ka mea i ka makaukau ana o "Enalapril" puʻe 'ana e loli ai i ka functioning o ka CCC, a me ka helu o nā nenoai i loko o ke kino, i kona hoʻokuʻu mai keʻena kūʻai lāʻau lapaʻau hana e kuhikuhi.

Helu 'o ka manaʻo a me ka pono o keia k e kaupalena' i 3 makahiki, mai ka la aku o kona? Iecaianoaaiiuo. Penei na papa io mai e lilo aku i ko lakou pākōlea waiwai ka wā waiho waho rula. Manufacturers Paipai 'ka malama ana i ka medicament i ka maloo, palekana mai ka pololei Map, i ka wela o ka ole e emi malalo o 15 a me ka ole oi aku mamua o 25 degere.

Analogs "Enalapril" i ka ia waiwai, no laila, koi pili ana i ka lāʻau, a me ka hiki ke mālama i kā lākou waho pūnaewele.

Pharmacodynamics medicament

Enalapril maleate (ʻeleu 'Oponopono papa) e iho, aole ia e pili i ke kaʻina hana i loko o ke kanaka kino keʻano o ka hanaʻana. Ka mea i keia hui ua manaoia e lilo i kekahi ano o ka "prodrug" i mea he hopena o ka uuku helu o ka hydrolysis reactions ho okumu i ka loa hou waiwai - enalaprilat.

He He e kaumaha ana ia ma luna o ACE ha awina ma mua o ka hoʻonāukiukiʻana o ka nui emi i loko o ka nui o ka aldosterone i loko o ke kanaka kino. Ma pōkole, i ke kanawai o ka "Enalapril" ninoieo i hookuu iho ke koko, (nā diastolic a me ka systolic) a me ka hōʻemiʻana haawe ana ma luna o ka naʻau Muscle (myocardium).

E like me ka hopena, lōʻihi-manawa loina mākou i loaʻa mai ia, hoʻowahāwahā i ke ka ho'ēmiʻana i loko o ke koko, ma hope o kona lawe ana i ka lāʻau "enalapril" nā mea maʻi i Ua i nele o ka nui o ke koko holo i loko o ka lolo. Eia kekahi,? Eaia papa hoʻokāʻoi i kaʻaʻa puʻuwai a me ka coronary koko pele.

Lōʻihi-manawa hoʻohana ana i ka lāʻau 'hōʻike kiʻekiʻe hopenaʻoi loa i loko o hypertrophic'aʻaʻa, IIeEeAIEUIeXAIIUE ma ka ventricle hema o ka naau Muscle, ma mua o kōkua e pale aku i ka holomua o ka naau ole. Eia hou, i ka Inc "enalapril" no 6 mahina, e hoʻoikaika i kaʻano o nā mea maʻi me ka hema ventricular dilatation a Circulatory kāna hana i loko o ka myocardium, mai ana ischemia.

Kaʻeleu lāʻau waiwai ua loaʻa i loko o ke koko, wai koko ma hope o 1 hola hope? Eaia o ka papa, a ma hope o 4-6 hola ihoiho kona i kā mākou. Ke hypotensive ia mau no i ke 24 hola.

ʻO ia pharmacological waiwai a me ka noho analogs "Enalapril" o ka hana hope.

Pharmacokinetics

E like me kūkā luna, omo o ka mea hana lāʻau waiwai i wahi lawa koke. Ke kemu wale ma kahi o 60% o ka enalapril maleate, ka buke kūpono kou holoʻokoʻa e hoopaa ana i ka wai koko nā polokina. Hoʻomalu huki nā mea kūʻai mai 'noonoo i ka mea i ke omo o ka hui mea i kalele iho ma ka aiʻai ana.

Ke kiʻekiʻe anal uku o ka enalapril ma-GHB nā pale kaʻa aie i ka hakakino 'ole o ka hana' Oponopono. No hoi ia mea hiki ke lanakila i ka placental ke'ākeʻakeʻa mai, a ua loaʻa i loko o ka umauma'aʻaʻa a me ka umauma waiu ma lactating wahine.

Excretion o ka lāʻau ua lawe maiʻano nui ma nā puʻupaʻa (60%). Ke'ōlelo mai ua hoʻololiʻia e hōʻike 'ia ma kahi o 20%, 40% - like me ka metabolite. I koeʻeleu waiwai mai ma ka naʻau liʻiliʻi, ai ka lākiō o ka enalapril / enalaprilat i nā hoailona 6-8% / 25-27%.

Nāʻikepili a me contraindications

ʻO nāʻikepili no ka hoʻohanaʻana i ka medicament "Enalapril" mea he paakiki mahuahua i loko o ke koko, kena ae la ia e maʻi e like me scleroderma a me ka CHF. Eia hou, i ka lāʻau ua pinepine hoʻohana 'ia i loko o prophylactic Inc i loko o nā mea maʻi me diagnosed coronary ischemia, haʻalele ventricular dysfunction (me asymptomatic). E like me lakou nei i ka lāʻau "enalapril" nāʻikepili no ka hoʻohana, akā, i ka pakiko-lapaʻau ma kekahi hihia ua i paipai. Wale i ka hoʻomalu hiki e i ka pololei lapaau regimen, a e hooholo i ka laʻau heluna.

Iloko o keia hookolokolo ana, ke kauka e no hoi e hiki ke hookupaa aku i ke alo a me ka wa e kaawale aku o ka hiki contraindications. Mau nā maʻi a me kāna hana o ka functioning o nā loko:

  1. Mahuahua pā lonoaʻili i ka hana 'Oponopono o ka lāʻau (like i "Enalapril" i ka ia manawa makemake no hoi e ana, e like me ka mea, i loko o ka hapanui manawa like i keia k hoʻomanaʻo).
  2. Hāpai keiki, lactation a me na keiki ma lalo makahiki 18.
  3. Previous hihia angioedema i lapaau hoomakaukau ana, mai ka pae ana o ACE-nā mea kūpale.
  4. Cerebrovascular insufficiency, a me nā cerebrovascular maʻi.
  5. Cerebrovascular hematopoiesis.
  6. ʻaʻa puʻuwai maʻi, me kaʻaʻa puʻuwai artery stenosis (unilateral aʻeluaʻaoʻao),ʻaʻa puʻuwai ka hoʻokō 'ole, i ke alo o ka transplanted hui,.
  7. ake maʻi.
  8. Maʻi o ka gastrointestinal'āpana, pu ma ka diarrhea a me ka luai.
  9. Scleroderma a me nā autoimmune maʻi ka heluna i ka connective nā'aʻaʻa.
  10. 'Aʻe' ana o metabolic keʻano o ka hanaʻana i loko o ke kino, a me ka hyperkalemia.
  11. Mimikō mellitus.

Komo "Enalapril" i loko o ka wahi, i hiki a pau i ho'ākāka 'ia ma luna pono e hoopau ia, a ua lawe Inc mai ma lalo o ka ikaika nā limahana o ka hoʻomalu.

Ka lāʻau "enalapril": i ka papa inoa o kaʻaoʻao loa

Ma naʻe o ka pomaikai nui o ka lāʻau, i ka wā o ka hiki aku o nā mea maʻi i 'ike i keʻano o kaʻaoʻao' ole e aloha ia Aneane pau hui, nenoai. Information ma adverse hanana ua loaʻa ma loko o ka papaʻaina ma lalo nei.

Adverse naoh i lalau i ka lāʻau

Nā loko, a nenoai

ʻaoʻao waiwai

Pinepine paha kekahi manawa

kākaʻikahi

Circulatory kahua

Excessive hakumakuma ke koko, palpitation, Orthostatic hypotension.

Arrhythmia, me tachycardia a me ka bradycardia, umauma eha, myocardial infarction, angina, pulmonary embolism.

alimentary kahua

A manao mai o dryness i loko o ka waha, epigastricʻeha, belching, nausea a me ka luaʻi, diarrhea paha constipation.

na naau oʻu iaʻi, hepatitis a me jaundice o pancreatitis.

Ka urinary'ōnaehana

Loli ma ka hakuʻala kuleana pili i, proteinuria.

______

ko mākou hopohopo kahua

Headaches, pōniuniu, luhi.

Syncope, Kanikani'āʻula, drowsiness, kaumaha, a mahuahua nui ko mākou hopohopo pīhoihoi a me ka iini pae, hilahila.

makaukau no

Tinnitus.

Hihia hoʻi ōhumu i loko o ka lewa, blurred hihio a me ka loli i ka pilikia makapō pokole.

naehana hanu

Runny ihu, nui puʻu, he lōʻihi manawa i maalo ae la oia i ka cough maloo.

Bronchospasm, pneumonia (interstitial).

Skin a me nā allergic reactions

Rashes, hives, angioedema i loko o ka poo (me mucous membranes o ka waha a me ka puʻu), ka ohane, erythema (me Steven-Johnson ka maʻi pale), likeʻole ano o ka dermatitis.

Pemphigus (vesicular poʻe noʻonoʻoʻole), Lyell maʻi pale, myositis, arthritis, arthralgia, glossitis, serositis, photosensitivity, vasculitis, atopic stomatitis.

Loli ma ke kumu o ke koko a me nā keʻena hoʻokolohua Eia kekahi laʻana

Hoomahuahua ae la lakou ESR, mahuahua lehulehu o ka urea i loko o nā Eia kekahi laʻana, hyponatremia a me ka hyperkalemia.

Hoonuiia ha awina o transaminases (hepatic), ua hoʻemi hematocrit, agranulocytosis, eosinophilia.

Other

"Iʻa", ua hoʻemi libido, Patchy lauoho me keia poho.

Kuhikuhi mauʻike manaʻo hoʻonāukiuki aku ma ka pololei keiki ma ke kino ka papa kuhikuhi hana lāʻau waiwai "Enalapril". Analogs (olelo ao no ka hoʻohana ana i ia na ike piha ma luna o ke kumuhana) hiki no hoi i like kāna hana. Ke ahonui, a me kona kauka mea nui, e hai i ka hoailona o kaʻaoʻao waiwai, e like me ignoring ia ke alakai i nui ka haunaele ma ka functioning o ke kino.

Pehea e lawe i ka papa "enalapril": ki ina hana like a me ka laʻau heluna

E stabilize ke koko, hoʻomalu waiho aku lōʻihi-makahiki hoʻohana ana i ka lāʻau '(me analogues a pau, no ka laʻana, "hexane Enalapril" lāʻau). Ma ka loiloi mua ke kahua o ka iapaau ana o ka hypertension ka mea, ua waiho, e lawe i ka lāʻau ma ka mahele lāʻau o ka 5 mg no ka lā. Ke kahua hoʻonohonohoʻana mahuahua ana o ka puʻe i ka elua pule o ka Inc ka laʻau heluna ua mahuahua ka 5 mg. He waiwai 'ana i kumumanaʻo ka mua 2-3 hola ma hope o ka hoʻomaka' ana o ka lapaʻau, e ia i ka hoomanawanui ma lalo o 'inikua hooponopono. Kēia kōkua e hōʻikeʻaoʻao 'ole i loko o kā lākou ulu. ʻO kā mākou mahele lāʻau E i oi aku mamua o 40 mg i ka lā, akā, i ka hoʻohana 'ana i ka nui o ka lāʻau mea hiki wale ina loa nō a me ka kupono tolerability o ka medicament.

Mahope o 2-3 pule ma hope o ka hoʻomaka 'ana o ka monotherapy "Enalapril" lāʻau, e hoolilo nā mea maʻi i ke kākoʻo lāʻau? Eaia? Aaeei. I loko o kēia wā, ke kela la i keia mahele lāʻau mea 10-40 mg lāʻau. Papa Pono e inu 1-2 manawa i ka lā. Paipai i lapaʻau mau ana ke koko,.

Ka mea ma luna o nā manaʻo paipai pili i ka poe e hoomanawanui i ka poe e ole e ae mai ka concomitant maʻi e like me hyponatremia a me renovascular hypertension. Ma ka nā māhele ka mea, e lawe i ka waiʻona? E like me ka rula, e hilinaʻi nui ma luna o na ano kanaka o ke ahonui, a me ka nui o ka maʻi. Ka loiloi mua mahele lāʻau i loko o kekahi hihia hiki ke ho omaulia wale ma ka hele kauka.

Duration o? Eaia o ka medicament hilinaʻi nui ma luna o kekahi mau aʻe, a loaʻa i ka hoʻomanawanui ka ana a me ka hopena o ke keʻena hoʻokolohua ho'āʻo ma. Mau loea, e hoailona oukou i ka abrupt withdrawal o ka lāʻau i alakai i ka io hopena. Nolaila, a hiki ina excessive hakumakuma o ke koko, i loko o ka hoʻomanawanui iki mai ka loaa ana i ka lāʻau "enalapril" E ke kiʻekiʻe o emi i ka laʻau heluna.

Symptoms a me ka lapaʻau o ka lāʻau overdose

No laila, nānā mākou i ka walaʻauʻana ano o ka lāʻau "enalapril" (papa), mai a ka mea kōkua, a me ka hopena o ko lākou? Eaia i loko o ka hopena. Ua ka manawa e neʻe ana i ke kūkākūkā o keia ninau, he overdose o keia k. Pinepine hoʻomanawanui iki mai kamaʻilioʻana, e lawe nui nā māhele o ka ai 'ma ka manaolana o ka pakele o kaʻawaʻawa loa symptoms. Ma ia hihia, ina e hana e lawe ka lapaʻauʻia "Enalapril" kanaka, i ka hopena hiki ia mea nui. Me ka ka ho'ēmiʻana o ke koko,'opi kānāwai i loko o nā mea maʻi i pinepine ana hiki aku ai i ka mea myocardial infarction a cerebral holo kāna hana.

Nō kāu, o ka mua symptoms o overdose i lilo o ka ike paka i, i ka noho ana o, nanea ana paha i keʻano o ke kāʻili 'ana. No hoi, aole e e hoi na hana mana o ka lesion o ka cerebral koko a me ka cardiac abnormalities: paleʻili, loa headache, eha ma ke kua o ka breastbone.

Lapaau o ka hoʻomanawanui me ka overdose o "Enalapril" symptomatic ka lapaʻauʻia. I ka mehana kaʻapu kōheoheo ua hōʻike loaa ana Saline a me gastric lavage. I hou loa na hihia i koi intravenous ka pahu kui o ka Saline a me ka wai koko ae pani ai, e like me hemodialysis.

lāʻau hana kūleʻa

Papa "Enalapril" hiki ke hana atypically, oiai o ka hiki aku a me nā lāʻau. Nonsteroidal Anati-hoʻoʻino ai '( "Ibuprofin" a me ka m. P.) A estrogensoderzhashie ai' pili kēia ho'ēmi i kona hypotensive hana. Blockers, nitratsoderzhaschie ai ', anesthetics a me ethanol hoomahuahua i ka hopena o ka lāʻau "enalapril". Diuretic ai 'i lawe pu me huaale i lalo, puʻe, hiki i hyperkalemia ulu. Me ka lōʻihi mālama nui e e lawe ia ai 'o ka pae mai o immunosuppressants, no ka mea, ma ka mea ami? Eaia me ka laau i loaʻa ka enalapril me ka nui loa ka hōʻoi' kona haematotoxicity.

ka lapaʻauʻia Reviews

I ka lā e pili ana i ka lāʻau 'hiki ke lohe nā maikaʻi a me ka io manaʻo. Ka mea mua nui ia Morohiha o "Enalapril" huaale - ke kumu kuai (20-25 rubles no pack) i ole e wahi hiki i ka mea kiʻekiʻe. Eia hou, nui mahalo i loko o ka makaukau a me kona laulā. Ke kūlana o ka papa kuhikuhiE drawbacks i ka nuiʻaoʻao reactions, a me ka pilikia kiʻekiʻe o complications ma ke alo o concomitant ka maʻi.

Ka hapanui o nā mea maʻi 'Enalapril' huaale kokua kiʻi pohaku uinihepa, o ke kahua hoʻonohonohoʻana mahuahua i loko o ke koko,. No nā mea kūʻai mai, ka poe i ko lakou hookohu ia ua kena ae la o ka haunaele ma ka functioning o likeʻole nā loko, ka mea, i ka haawi mai i wale ma luna o ka lāʻau, akā, no hoi, mai kona analogues, e like me ia ma ka hapanui o na hihia, ka mea iloko o ka iaʻeleu waiwai a me ka e like enalapril indapamide. A no ke aha la poe akamai i ka mea,ʻaʻole loa waiho aku e lawe mau ai 'lakou ma ke koko,.

Analogs "Enalapril": na oko, pono a me keakea

Ma neia manawa, ua nui loa ai 'ana e like me ka lāʻau "enalapril" ke ao nei mea lāʻau lapaʻau market. Loa pinepine, ka mea, i ka oi aku waiwai e lilo aku, i 'aʻole i mau kumu i ka wa e kaawale aku o adverse reactions a oi aku lāʻau hopenaʻoi loa. E noonoo i ka papa inoa o ka ai 'ana i haku o kaʻeleu waiwai, like me ka mea i loaʻa ma loko o ka "Enalapril" papa. Nō kāu, o ka mea lāʻau lapaʻau keʻena hoʻokolohua ma Western aina ua hoʻohana 'ia e like me ka papa kuhikuhiE ke keʻena amplodipin enalapril, i ÿokoÿa o enalapril maleate mea wale nō i loko o ka hakakino' ole. I ole ia ka mea, i ka ia 'ano a me ka waiwai.

Ma ka Lūkini mea lāʻau lapaʻau market ma laila nō nā kēia mau analogs "Enalapril":

  1. Papa a me nā capsules no injectable "Enap" ma Kolewenia poe KRKA. Lākou kumukuai hoomaka ma ka 280 a me ka pii ana ae i ka 4000 rubles no ka'ōpala o ka papa, a me ka 500 rubles no 10 ehiku huewai i ka pāʻoihana. I hiki ke ike, ma ka Akä naÿe i ka "Enalapril" lāʻau, i ke kumu kūʻai o he kiʻekiʻe, aʻo nā huahana o keia momoku ahi inaccessible i ka helu nui o nā mea kūʻai mai. I ka Ia manawa, poe akamai i nana i ka mea kiʻekiʻe ma Hawaiʻi o ka Analog.
  2. Papa "Enalapril hexane" mai ka German Hookah SANDOZ. Wahi lulu lāʻau no kona laulā mea i emi iki mahope o ia i ka haawiia mai medicament. Ke kāki o ka mea like, ke'ōlelo mai iki ma luna ma mua o ka uku o ka "Enalapril" a me ka mea e pili ana i 78-100 rubles no pack.
  3. Papa "Berlipril" hua mai la ia e Kelemānia mea lāʻau lapaʻau poe, "Pelelina-Chemie". I ka papa kuhikuhiEʻeleu 'Oponopono o ka lāʻau mea amlodipine, enalapril. Aie i ka mea i ka loaa ana o ka hui i oi huikau a me ka pipiʻi, papa kāki mea e pili ana i 140-180 rubles no pack.
  4. Papa "Renitek" mai MERCK, ke kumukuai o ka i mea he iwaena konu o ka huahelu a me ka mea 80-150 rubles no pack.

Nō hoʻi i loko o nā keʻena kūʻai lāʻau lapaʻau 'oe e huli i na like me ka' ole a me ka hoʻokō 'ana i ka lāʻau' analogues "Enalapril" like "Kalpiren", "Miopril", "Envas", "Vazopren" a me ka "Miopril". Poe akamai, nae, e olelo aku i ua ole mau oleloia ai 'hiki ke hoʻohana i ka hope i ole kokoke i ke ahonui, no ka mea kumu, na wahi lulu lāʻau. Ka mea o ia i loko o kona haku mele 'ana ka mea, kokoke haʻi hou aku mākou "Enalapril", a' o ia hoʻi i ka mea hiki no hoi i keʻano o nā complications. Nō hoʻi, ua aʻo aku ai iā kauka, e hoʻolohe i ka haku mele 'ana i lawe wale aku lāʻau. Amplodipin enalapril, i ÿokoÿa o enalapril maleate mea uuku, e hiki no hoi ia hana he kūlana ma ke kino. Ma kekahi hihia, mamua, e hoʻohana i ka iniiaiie lāʻau o kekahi o na hua analogs, ia mea pono, e kukakuka pu me ke kauka.

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