Ola kino, Hoomakaukau
"Formetin": aʻo no ka hoʻohana 'ana, maoli
Currently mākou i loaʻa hou kanaka me mimikō a me na complications o obesity type. He nui ai 'loaʻa no ka iapaau ana o kēia mau maʻi puʻuwai. Kekahi o ia mea i ka laau "Formetin". Kona salient hiʻona e e wehewehe i loko o kēia 'atikala.
mea lāʻau lapaʻau waeʻano
"Formetin" kauoha no ka hoʻohana i ka hōʻike i loko o kēia 'atikala, mea he biguanide hypoglycemic lāʻau pae.
Description o ka haku mele 'ana a me ka hoʻokuʻu ke ano
Ma kekahi o kona papa.
m, g. | m, g. | m, g. | |
Kaʻeleu 'Oponopono | |||
metformin hydrochloride | 0.500 | 0.850 | 1,000 |
kākoʻo 'ona | |||
povidone waena hakakino type | 0.017 | 0.029 | 0.034 |
croscarmellose paʻakai | 0.008 | 0,0136 | 0.016 |
makanekiuma stearate | 0.005 | 0,0084 | 0.010 |
Available lāʻau "Formetin" ma ka blisters 100, 60 a me 30 o na papa io.
Waihoʻoluʻu White maloko o na papa a me ka laʻau heluna palapala hilinaʻi nui ma luna o ka waihona ipu mea. Ma 500 mg ploskotsilindricheskoy ka mea, i ka hoʻopoepoe kinona me ka hoailona, a chamfered. Nō hoʻi ka laʻau heluna o 1000 mg a 850 mg i "Formetin". Nā papa ma keia hihia, convex a me ka'ololaha. Ka mea, i hoʻokahi-kapakahi kamepiula.
pharmacodynamics
Metformin ( "Formetin") 'aʻole hoʻi gluconeogenesis e kahe ana i loko o ke ake, a pela he mea he emi ma ka glycogen hale kūʻai ia. Kēia mea kökua ka poʻea pau i ka pilikia o ke omo mai ka intestinal monakō koko, ka hōʻoi 'i ka wehe' ana i ke koko kō pae o ka'ōnaehana. Kēia maoli i ka pane o nā'aʻaʻa e insulina me ka mea e pono ai ka? Iecaianoaaiiie o kona endocrine hapa o ka pancreas B-keena, piliwaiwai hypoglycemic naoh, no ka mea, ua i ho'ā '? Iecaianoaaiiuo o la waiwai.
Uluwehi O "Formetin" hōʻike manaʻo i olelo e pili ana i kona laulā, ho'ēmi i kā ka mea nui o ke koko i loko o ka "ino" naʻokoko a me triglycerides. Ka maʻiʻo o ka kiʻekiʻe nuʻa lipoproteins keia maoli he i 20-30%. Me ka ineffectiveness o kaʻai lāʻau "Formetin" kauoha no ka hoʻohana a ua ho'ākāka 'ia i loko o kēia' atikala kōkua e ho'ēmi a / a stabilize i ka hoʻomanawanui i ka hoʻokauʻana. Kēia ka hana aie i ka'okesaside o ka monakō koko ma o oxygen-noa, a emi kona'ōpū. Nō hoʻi ka mea, blunted'aʻaʻa plasminogen ho'ā hope kaʻina hana ma ka hana ma luna o kona inhibitor, ai ka hemostatic kanawai i Konakele.
Pharmacokinetics
Kaʻaluna metformin hoʻomaka ma ka gastrointestinal'āpana. ʻO kā mākou nui o ka waiwai i loko o ke koko mea e pili ana i 2,5 hola ma hope o ke noi i ka uku o ke omo pa alima mahele lāʻau - 50-60%. Omo mea e like ai o ka lāʻau i loko o ke kino e loli ai i ka pilina ma waena o kaʻeleu waiwai, a me ka kumuʻiʻo i loko o ka wai koko. I ka papa "Formetina" i pili i ka wai koko nā polokina. Ua olelo e pili ana i kona laulā. Mai ka uuku o ka paa ololi, ka lapaʻau ua maikai ke kemu. Palapala moʻopane o ka hakuʻala, akepaa, ma ka Muscle'aʻaʻa, ma ka salivary glands. Ma ke kino, metformin koe ua hoʻololiʻia. He a laila excreted ma nā puʻupaʻa. No laila, ma ka hihia o ka 'aʻe' ana o kā lākou hana ua malamaia hoʻomāhuahua. Liluwelo hapa-ola o 1.5-4.5 hola.
naue like
Medicine "Formetin" ua hoʻohana 'ia no ka iapaau ana o kekahi mau waeʻano o ka maʻi. ʻo ia, i ke alo o ke 'ano II mimikō, me ka obesity hihia a me ka huikau ka wā o kaʻai, aole ia i kōkua i ka malama i ke koko kō pae maʻamau, a hiki ma ka hui pu ana, me ka sulfonylurea. I ka hoʻokō o ka "Formetin" no ke kaupaona poho.
Pehea e lawe?
Ka mahele lāʻau o ke kauka 'o ia hoʻi Nāna e koho, ma muli o ka nui o ka monakō koko i loko o ke koko. Una aaieieno? Mea pono ke hana ma hope o kaʻai, e hui pu ana me ka nui o ka wai a me kaʻilikai i ka papa machining. Me ua i haiia ae maluna, i ka laʻau heluna ua hoakaka ia ke kaumaha ma muli o ka maʻiʻo o ka monakō koko i loko o ke koko. Ua hoʻomaka me ka palena iki nui - 0.5 g. A 0,85 g. No ka lā. Mau lā e hoʻomaka ana lapaʻau me keia k ma hope ua lilo i ka napoo ka maʻiʻo o metformin i loko o ke koko. Kohoʻia, ke kiʻekiʻe o mahuahua ka mahele lāʻau a kekahi i kā mākou waiwai. He like ia 3 nā huna.
Mai ka kūpuna pinepine malama i ka hooulu ana o lactic acidosis, no ka ia i ka nui o ka mea i kā mākou i kela la mahele lāʻau o ka 1 g. Nui o ka lāʻau ua i hoemi ma ka 'aʻe' ana o pūnao, i mea e pale aku i ka allergic naoh, i hoike mai ai ia ia iho i loko o ka palapala o ka ili rashes, a me nā mea hiki adverse hanana, a e e hoakaka ma lalo nei.
Contraindications
Ma keia manao, he nui na nuances. Uluwehi O "Formetin" kauoha no ka hoʻohana i ka hōʻike i kēia kikokikona, ua contraindicated ma ke alo o ka:
- Diabetic ketoacidosis, precoma, coma.
- Loa hihia hoʻiʻaʻa puʻuwai functionality.
- Cardiac a me ka ÷ naehana hanu ole.
- Huʻi pae o myocardial infarction.
- Dehydration.
- Maʻi alcoholism a me nā kumu i ke hoʻonui i ka hoike ana o ka ulu lactic acidosis.
- Huʻi hahau ana.
- Hāpai keiki, a breastfeeding.
- Hypersensitivity i keia srudstvu.
- Majorʻoki kino a me ka poino, insulina ua hoonohoia ka wā.
- Loa infectious maʻi.
- Ooieoeiiaeuiuo kāna hana o ke akepaʻa.
- Huʻi waiʻona kaʻapu kōheoheo.
- Lactic acidosis (me mōʻaukala).
- Hypocaloricʻai (emi o 1000 kcal. Per lā).
- Adioizotopnyh a radiographic haʻawina, i ka hooko ana o ka waiwai iodide type.
Ua ua no hoi e waiho i ka hoʻohana i ka lāʻau "Formetin" kanaka no makahiki he kanaono, ae hana i kāohi, ua koi ikaika hana. No ka mea, i loko o keia hihia, ka mea, i ka māhuahua pilikia o ka ulu lactic acidosis.
ʻaoʻao kanawai
Ka hanana o ia kaʻawaʻawa loa symptoms me "mea hao" ho'āʻoʻana i loko o ka waha, ka luaʻi, nausea, diarrhea, flatulence, nele o ka ikaika loa ka makemake pono discontinuation o ka pono o ka lapaau a me ka koke kōkua i ka hoʻomalu. Lōʻihi-manawa hoʻohana ana i ka lāʻau 'ke kumu o ka haunaele a piha cessation o kaʻai ana o ka wikamina B 12, i hiki aku ai i ka hoʻomāhuahua i loko o ke kino o ka la mahope, ma o na la wikamina ia wā. Ma pohihihi keia hoopii, ulu aʻe - megaloblastic ka 12-hiki ole no ia anaemia. Inā improperly lawelawe mahele lāʻau hiki hypoglycemia. E hiki no hoi ka mahina allergic reactions e like me ili wikiwiki. No laila, i ka lāʻau "Formetin" hōʻike manaʻo a ma luna o kona appropriateness ma o ka hoʻohana 'ana o kekahi, E e hoonoho wale ma ka hele kauka.
Cautions
An nui hiʻona i ho'ākāka 'ana hoʻohālike ho'āhu kumu waiwai "Formetina" ma ke kino, a me ka ia mau hopena o keia.
E pale ai hoʻomāhuahua o lactic acidosis a me ka Kāohiʻana o ka metformin, ia mea pono ke kanaka hoʻoponopono i nā nā hoailona o ka hakuʻala hana, a no ka ho'āʻo e hooholo i ka maʻiʻo o lacticʻakika i loko o ke kino ma ka liʻiliʻi 2 manawa no ka makahiki. No hoi, ina oe i eha ma na nāʻiʻo e e retested.
Ke kanawai o ka la lāʻau ma luna o ka hana, e kipaku aku maomeka, a kipaku kaa
Ma keia hihia, e like me ka mea, i kekahi nuances. Hopena "Formetina 'hana i ka hana a me ka hana amo i wahi wale ina ia i loko o ka huipūʻana me ka ai' ka heluna i ka hana keʻano o ka hanaʻana i kauoha i ka mämä holo o ka pane, a mahuahua lehulehu. He nui ka ike.
Noi o ka hāpai keiki, a breastfeeding
E hoomakaukau ai "Formetin", kuhikuhi no ka hana ana i ua ho'ākāka 'ia ma keia, i' ole ma o ka fetus waeʻano «B» e FDA. Ma hāpai keiki ke loaa i kēia kālā. Eia naʻe, kona hoʻohana hiki e wale i loko o kekahi mau hihia. O - ka wā manao hualoaʻa mai keia Inc, e oi aku i ka loaʻa nui o ka Loaʻaʻia kamepiula a hiki i ka fetus. I Kekahi Mau a me ka hihia haʻawina ma ka hoʻohana 'ana o kekahi mea paahana e like me ka lāʻau "Formetin" i alakaʻi i ka wā o ka hāpai keiki. I ka manawa o ka iapaau ana e hooki breastfeeding. Ma kekahi hihia, e pono e nīnau aku i ka palapala hōʻoia no kauka.
lāʻau hana kūleʻa
Metformin maoli i ka nui o ke koko kōpaʻa. Keia mea pakahi aku la ia mea i ka i ka wā hoʻokahi? Eaia o ka pili-steroidal Anati-hoʻoʻino ai ', sulfonylurea nā mea loaʻa a me ka clofibrate, monoamine oxidase nā mea kūpale, acarbose, insulina, oxytetracycline, cyclophosphamide, nā mea kūpale o angiotensin hoʻololi''ūhū blockers a me type.
I ka pili pu me endocrine ai '(ku una ha contraceptives, corticosteroids, sympathomimetics epinephrine, thyroid gland hormones, glucagon, thiazide a "loop" diuretics, phenothiazine nā mea loaʻa, nicotinicʻakika nā mea loaʻa) e metformin hypoglycemic ke peleki pāʻana kaʻina.
Me he huihui 'ana o ka mea paahana e like me ka lāʻau "Formetin" me "Tsimidinom" "nifedipine" ulu pilikia o lactic acidosis, metformin inhibiting ka excretion mai ke kino. Oia mālama i loko o ka hana o ke kanakaʻona mau huahana, ma ka Vol. H. Ma ka haku mele 'ana o nā lāʻau.
Cationic konohiki (quinidine, amiloride, digoxin, procainamide, Morphine, quinine, vancomycin, ranitidine, triamterene) i hanaʻia i loko o nā tubules, vying no ka amo'ōnaehana a me ka lōʻihi-makahiki lapaau e hoomahuahua i ka nui o ka lāʻau lehulehu i 60%.
overdose
Overdose "Formetinom" ka wā lawe 0,85 nā huna no ka lā, a hoʻonāukiuki lactic acidosis malama. Nō hoʻi, he kiʻekiʻe ka maʻiʻo o ka metformin hālāwai hoʻolohe i ka hakuʻala ole.
I kakahiaka nui symptoms o lactic acidosis i ka nawaliwali o ke kino a pau, bloating, haʻahaʻa kino mahana,ʻeha i loko o ka opu a me nāʻiʻo, ma lalo ke koko, reflex bradyarrhythmia. Ma kekahi mau hihia, ma laila nō pinepine hoikeana o naehana kāna hana, pōniuniu, a, me ia i kaʻilihune, he mea no ka hooulu ana o coma.
Ma ka mea iki o ka symptoms o overdose e ka hoʻohana 'ana i ka lāʻau' ana a me ka nīnau aku i ke kauka e hōʻoia i kaʻike, o lactic acidosis. No ka wehe 'ana o ka mea hana waiwai o ka Agena, a lacticʻakika, mai ka meaola e hemodialysis laua me symptomatic lapaau.
"Formetin": counterparts
Aia nō he wahi lihi iki o ka waiwai o kēiaʻano. Analogues "Formetina" nei iluna mea haʻilula keimikala i loaʻa i loko o kona haku mele 'ana e like me ka papa kuhikuhiE ke keʻena o ka metformin hydrochloride. Kekahi laʻana o ka lāʻau o Lūkini nā hoʻohua, "Vero Metformin," "Gliformin", "metformin", "Metformin-Richter", a me ka huakaʻi i ke kai - "Glucophage", "Glucophage" a me ka "Glyukofazh Long" (Farani), "Lanzherin "(Solowakia)" Metfogamma "me ka loli iki ana dosages oʻeleu waiwai o 0,100, 0,500 a 0,850 g. (Germany).
Nā kūlana a me nā hua'ōlelo
Ma keia manao, eia kekahi mau rula. E hoomakaukau ai "Formetin" mea he potent, pela no ka mea, ua hookuu wale ma ke kuhikuhi a me ka pono waho pūnaewele i mehana ea, mai o ka loaa ole mai o na keiki a me Map wahi. Holopapa ola ia - 2 makahiki.
kāki o
Ka awelika uku no ka lāʻau "Formetin" ua kau ke kaumaha ma muli o ka laʻau heluna mai ka 59 rubles. 0.5 g. O ka blister, 133 rubles. o 0,85 g. a me 232 rubles. no 1 ka makahiki
ka hopena
A pau ka keia ka loaʻa o ka hailonaʻana no maikaʻi kēia 'ike. heluhelu i kēia 'atikala ma hope, kela kanaka keia kanaka e e hiki i pane i ka ninau o ke ana, e lawe' Formetin "a me ka mea ia i ka waiwai, e imi.
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