Ola kino, Hoomakaukau
Ka lāʻau "Celebrex": hōʻike manaʻo, analogs, aʻo no ka hoʻohana 'ana, uku
I ka make ana o ka spine, hanahana loa kaʻeha ma na ami a me ka connective'aʻaʻa loli oihana ma luna o ke kāʻei kua o ka li nui - Eia naʻe, i kēia mau maʻi e noho ana i ka loa, he pono ole i loko o kā mākou manawa. Ma keia wahi o ka mea e loli ai I Aloha Hawaii, nele i ka kino ai haʻawina, aaiaoe aʻe. Ma waho aʻeo i ka loa eha i kanaka e ae aku ana ma keia ano, maʻi hiki no e luku mai i ka pau meaola, hoololiia'na koko kemika a me ka heluna o ka maʻamau functioning o na nā loko.
He nolaila, nui ke kanaka hoʻoponopono i ke ola a me ka manawa e pono i ka maʻi. Kekahi o ka loa ka hoʻokō ai ', a no a hiki i ka pae o ka ole-steroidal ai' kapa medicament "Celebrex". Reviews o nā kauka e hooiaio aku kona laulā ma ka like ana me ka laina hookahi o Anati-hoʻoʻino ai '.
I ka papa kuhikuhiE hopena o ka lāʻau
Mea pomaikai o ka lāʻau i ke kapaʻia kona hiki e inhibit i ka hoʻoʻino kaʻina ha awina ma kekahi mau kahua o ka hoʻonaʻauao o ka maʻi. Noho i loko o ke koko, i ka lāʻau mea hiki ke inhibit TSOG2 kaʻina e hiki aku ai i ke ola o ka li nui. "Celebrex" ka lāʻau i ka ikaika analgesic waiwai antipyretic haʻawina. Nolaila, ia eliminates ole wale i ka li nui foci, akā, i hoʻi mai kēlā wahi e lawe aku oe i ke koʻikoʻi eha, ho'ēmi i kā kuni.
Nā pono o kēia huahana nā kona ka palena haʻahaʻa kanawai ma ka platelets, i mea, i ka lāʻau 'aʻole ole i pilikia i ke koko clotting. Ka wā e loaʻa mai i ke pili-steroidal Agena i ka mea, aole ae hookaawale ana i ka opu a me ka naʻau liʻiliʻi, hoemiia ka pilikia o ulcers a me gastritis nā mea maʻi.
No laila, e hoʻohana nui aku i lohe nui i ka "Celebrex" huaale ma mua o nā NSAID ai ', "naproxen", "Aspirin", "ibuprofen".
directional
"Celebrex" capsules i ka hiki e ho'ēmi i ke oolea o ka hui eha, oolea hoʻopau ia Makuakane me excessive nani. Oia waiū hiki, e pono e hoomanawanui i diagnosed me rheumatoid arthritis, osteoarthritis. Kanawai o ka lāʻau 'ino i ka mea i kā mākou hopena ua 24-48 hola ma hope o ka mahele lāʻau mua. Dysmenorrhea lāʻau kuleʻa eliminates ka eha, a me ka loa huʻi. No hoi, ka mea, ua pono ia no ke kokua o ka eha ma hope oʻoki kino (maxillo-lehalehu, a orthopedicʻoki kino).
Nā mea maʻi me ka ankylosing spondylitis lāʻau "Celebrex" hookaaokoa ae mai o ka pathological keʻano o ka hanaʻana, a hoonui ae i ke kino o ka hana, e kuleana pili i. I ka malama ana i naʻano o nāʻohana adenomatous polyposis hoʻohana ana i ka lāʻau 'alakai ai i ka nui ka ho'ēmiʻana i loko o ka ulu ana o polyps ma ka AeXIeAaOIePEAaI a me ka duodenum: hoemi i ko lakou helu a me ka nui. Kauka koi i kūpono nā māhele o ka lapaʻauʻia a me ka adherence i ka lapaʻau regimens ke hoʻokō maikaʻi loa i nā hualoaʻa me ka hoʻohana 'ana o "Celebrex" lāʻau. E hoike hōʻike ka palena haʻahaʻaʻaoʻao 'ole ana e lawe i kēia ka lapaʻauʻia.
Ke kinona a me ka haku mele 'ana o ka lāʻau
Loa e wae inhibitor mea he gelatin mea hōʻikeʻikeʻuʻuku kokoke keʻokeʻo paha keʻokeʻo, ka mea mau i ka aniani moakaka, a ua hoailono aku la ia me ka uliuli holehole mai ai i 'ae' "7767" ma kekahiʻaoʻao, a "100" a me ka "200" ma o ka 'ē aʻe. Mea hōʻikeʻikeʻuʻuku Contents: granulated keʻokeʻo 'ia nā pōpō.
I ka haku mele 'ana o ka lāʻau nā: celecoxib (walaʻauʻanaʻeleu' Oponopono), lactose, povidone K30, paʻakai lauryl sulufahate, makanekiuma stearate, paʻakai croscarmellose. Ka iwi ua i ka titanium'okikene lua, a me ka edible gelatin. Inā kūpono hooponopono o ka lāʻau intramuscularly injections pau i waeia "Celebrex". Kēiaʻano o ka lapaʻauʻia ua hookuu ia ma ke ano o ka pāʻoihana no ka pahu kui o 2.2 ml ampoules - kumu waiwai celecoxib.
Pharmacokinetics
Ka lāʻau 'Ua pono paka i loko o ke koko i loko o ka hooke ai ana moku'āina, a me ka i kā mākou hana ma hope ma kahi o 2-3 hola hiki, naʻe, ka hoʻohana' ana o nā mea a pau me ka momoma ai e hoʻokaʻulua kona hoʻomāhuahua no ka 1-2 hora, No ia mea, ia mea e pono, e nīnau aku i ke kauka e pili ana i ka manawa o ka lawe i ka lapaʻauʻia.
Noho i loko o ke koko, i ka hana waiwai mai e hoopaa i ka ula koko keena, akā, i keʻano papa hana aʻole e pili mai ka e piʻi like ana o ka makemake lehulehu o ka lāʻau i loko o ke kino. Uluwehi O metabolized i loko o ke ake e'okesaside a me ka glucuronidation ke komo pū CYP2C9'ūhū. Ia auoiaea ia hoʻi, me ka mimi a me feces ma ke ano o ka poe noonoo ole metabolites, a me 3 wale% o kaʻeleu waiwai koe ua hoʻololiʻia.
Uluwehi O "Celebrex", analogues o ka i mea like me ka haku mele 'ana, loaʻa hoʻi, e kauoha ana ka palena haʻahaʻa pōʻino ke ola, ka hoʻopiʻi ai i kona hiki no e hoʻokemuʻia ma ka mea i hiki, a kokoke loa eliminated mai ke kino. Me ka haʻahaʻa kino kaumaha malama i ka lehulehu ma luna o ka lāʻau i loko o ke koko, a ua mālama aku ma mua o ka wahine keia kŰia. Ua uaʻAʻoleʻikeʻia ke kumu, akā, i loko o kanaka Naʻau malama i ka iaʻano. No laila, i kēia mau pūʻulu o nā mea maʻi i hoakaka ia i ka haʻahaʻa mahele lāʻau o ka lapaʻauʻia ma ka hoʻomaka o ke Inc.
nāʻikepili
E like me ka ole-steroidal Anati-hoʻoʻino Luna no ka symptomatic lapaʻau hoakaka lāʻau "Celebrex". Nāʻikepili no ka hoʻohana:
- rheumatoid arthritis;
- osteoarthritis;
- spondylitis;
- algomenorrhea;
- huʻiʻeha (kia-operative manawa, hoʻi eha, musculoskeletal maʻi);
- hoʻohana 'ia ma ka hana maikaʻiʻole o adenamotoznogo polyposis.
It E e kaulana i kūpono lapaʻau ke haawi wale i kekahi kauka ma ke kumu o ka noiʻi.
Nā Papahana O Ka hooponopono ana i ka lāʻau '
Lālau aʻela ia i ka lāʻau 'pono ia i loko, ka nānā' ana i ka palaoa. Chewable papa e ole e, e pono e inu akaka ka wai. It E e kaulana ia mea'ōnaehana mānowai koko complications ke'ākoʻakoʻa me ka maʻi hooponopono o ka lāʻau. Nolaila, kauka i hoakaka ia "Celebrex" He pōkole papa o ka lapaau. House poe akamai i hōʻoia i ka i kā mākou mahele lāʻau no ka lōʻihi-makahiki lapaʻau e ole oi aku 400 mg no ka lā!
- Lapaʻau o osteoarthritis - e pono mahele lāʻau mea 200 mg no ka lā. Chance o ka hookahi mahele lāʻau a mahae i loko o elua (ma ka pololei,ʻanuʻu).
- Rheumatoid arthritis - manaoia mahele lāʻau o 100 a me 200 mg no 2 manawa no ka lā. I ka wā o ka loa loa pepa - mai i 400 mg palua i ka lā.
- Ankylosing spondylitis - 200 mg no ka lā, no ka 1 a 2 māheleʻia nā māhele. I ke kauka o ka manao i ke mahuahua ka mahele lāʻau e pono ai
- Dysmenorrhea a me ka ikaika eha - hoʻomaka Inc me 400 mg no ka lā, a hui pu kekahi 200 mg i ka lā mua o ka Inc, ina he pono. I ka kēia mau lā, e pono e lawe 200 mg palua i ka lā.
Duration o ka iapaau ana me ka nānā 'ana i ka hele kauka.
Contraindications i ka hoʻohana 'ana i ka lāʻau'
Ma waho aʻeo i hiki allergic reactions i constituents o ka lāʻau, he mea kapu ma lalo hali 'ana paha ma ka hoʻohana' ana i ka lāʻau "Celebrex":
- Bronchial asthma, urticaria, allergic i nā NSAIDs.
- Ke postoperative wā ma hope aortkoronarnogo holo alaʻokoʻa.
- Peptic ulcer (exacerbation).
- GI kahe ana ke koko.
- Hoʻoʻino na naau oʻu maʻi.
- Heart ole.
- Loa hepatic insufficiency.
- ʻaʻa puʻuwai insufficiency.
- Hāpai keiki, a lactation.
- 'Aʻole i haawiia no ka hoʻohana ma lalo o 18.
- Hypersensitivity i na constituents o ka lāʻau a me ka sulfonamides.
Kaiapuni e hoʻohana i ka lāʻau me ka loliʻana i loko o ke kino, maʻi o ka mea'ōnaehana mānowai koko nenoaiu, mimikō.
ʻaoʻao waiwai
I loko nō o ka potency kiʻekiʻe o ka lāʻau, hooloihi ae i a pololei ole? Eaia 'ano a me ka laʻau heluna hiki eʻaoʻao' ole o ka lāʻau "Celebrex". E hoike hōʻike i ka loa, he pono ole (pinepine) symptoms e like me:
- Allergic reactions me ka poʻe noʻonoʻoʻole, urticaria, pruritus.
- Flatulence, dyspepsia, edema, Kanikani'āʻula.
- Cough, rhinitis, maʻi palū-me naoh a me ka ÷ naehana hanu'āpana nā mea palahēhē.
- Urinary'āpana nā mea palahēhē.
Ka emi ka mea, mahuahua ka iini, anaemia, tinnitus, flushes, arrhythmia, arterial hypertension. Kekahi nā mea maʻi i kākau ulceration o ka digestive'āpana, angionevropatichesky edema, i ke kahua o ka bullae ma luna o kaʻili, exacerbation o pancreatitis a me kona ulu ana, hilahila. hiki wale nō i kēia mau symptoms i hoʻomaka ai ka wā i ka papa o ka lapaʻau ka pokole (i ka 12 pule,ʻaʻole e oi aku 800 mg no mahele lāʻau). Akā, ma ka hihia o ka lōʻihi-makahiki lapaʻau (mai ka 3 makahiki) i malama:
- Common: hāʻule pohō wale o ka noho, hypertension, nā mea palahēhē o ka pepeiao, angina, myocardial infarction, nausea, dysphagia, prostatitis, mahuahua creatinine.
- More pohihihi keia: arrhythmia, angina, ischemic hahauʻana, atherosclerosis, hiamoe kāna hana, vaginal kahe ana ke koko, ulcers o ka waha, dysmenorrhea, māhuahua ma ka hemoglobin, emi ma ka hematocrit.
Ke AaOIeIOUIeXAOAaIN o ka lāʻau a me nā ai '
Ke medicament 'Imi biotransformed pili i P450 2C9 (cytochrome). He nolaila, e hiki pololei AaOIeIOUIeXAOAaIN o ka lāʻau a me nā konohiki:
- Concomitant ana o ka ai ' "Warfarin" maoli i ka pilikia o ka ona kahe ana ke koko.
- E hoomakaukau ai "Ketanazol" a me ka "Fluconazole" hoomahuahua i ka lehulehu o kaʻeleu waiwai celecoxib aneane papalua.
- Loaa ana blockers a ACE nā mea kūpale angiotenzita NSAIDs ke me ka nui loa ho'ēmi i kā lākou antigipertinzivny ai
- Me ka hui pu huahana i loaʻa ka likiuma, ka mea hiki me ka nui loa hoonui i ke koko pae.
- Ua ua papaia e ka poʻe hoʻohana i ka lāʻau "Celebrex" analogs i loaʻa ka celecoxib, nā NSAIDs!
lāʻau analogues
Ua mea waiwai 'ana i kumumanaʻo i "Celebrex" lāʻau koina i nui loa, kona kumukuai mea ma awelika mai ka 400 a hiki i 450 rubles. 10 capsules (100 mg laʻau heluna). Eia naʻe, ua lapaʻau mea nō pipiʻi no ka hoʻomanawanui i ka lōʻihi-makahiki Inc. Ma keia hihia, ke ae ole o ke kauka, hoonoho konohiki i loaʻa celecoxib. No ka lāʻau "Celebrex" analogues o ke kēia:
- lāʻau "Ranselak";
- lāʻau "Revmoksib";
- papa "Flogoksib";
- mea hōʻikeʻikeʻuʻuku "Artoksib".
Mau analogs pihaʻi me na iaʻeleu waiwai, a i ka kūpono kou'ālike pākōlea hookoia ma ka iapaau ana o ka maʻi. E noke ana no hoi ia he kūpono mahele lāʻau o ka mea like wale nō ma ka hele kauka. Ma keia hihia i ke kauka E hoomanao i kekahi haku mele 'ana kōkua iā ia, i loko o analogs, ka mea, aia no iloko olaila na mea hoʻonui i like i ka lāʻau "Celebrex". Instruction Nāʻana na kumu paipai i ka manawa kūpono o ka allergic naoh ma ka hoomanawanui i na excipients o kekahi mau lapaʻauʻia kekahi pae.
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