Ola kino, Hoomakaukau
"Paroxetine": aʻo no ka hoʻohana, nāʻana. lāʻau analogues
He aha ka mea i manaoia lāʻau "Paroxetine"? Na Ke Kumu no ka hoʻohana ana i ka lāʻau, e e hōʻike i loko o kēia 'atikala. No hoi kekahi poe mai o ia oe i ka ike o kekahi contra-nāʻikepili a i loaʻa mai i kēia ka lapaʻauʻia, ina loaa ia ia kekahiʻaoʻao waiwai, i loko o ka palapala i loaʻa, a pehea ka lāʻau hana me'ē aʻe ai '.
Haku mele 'ana, a me ka'ōpala ke ano o ka lāʻau kalaʻana
Uluwehi O "Paroxetine" hele i kuai i loko o ka palapala o ka papa, ho film-kapa komo iā ia. Ka mea, e hoʻopoepoe a me ka lenticular kinona, keʻokeʻoʻeleʻele, a me ka pilikia o ka hoʻonaninani ili.
Kaʻeleu waiwai ua noʻonoʻoʻia e mākou 'o ia hoʻi paroxetine hydrochloride hemihydrate. Nō hoʻi, i ka lāʻau i loko o kona haku mele 'ana, ua kākoʻo nā kumumea i loko o ka palapala o ka colloidal silikone'okikene lua, microcrystalline kelulose, crospovidone, kalipuna hydrogen posapahate, copovidone, talc a me ka makanekiuma stearate.
Papa "Paroxetine" i kūʻaiʻia i loko o blister he huihui 'ana o 10 apana a i waiho ia ma ka pepa pahu.
Ke pharmacological hana o ka lāʻau
He aha mea i ka lāʻau "Paroxetine", a analogues e kapaʻia he iki ae la, e? He he antidepressant. He he inhibitor o (e wae) serotonin reuptake lolo neurons. Kēia ka mea hoʻoholo kona Anati-depressive 'ole a me ka hopenaʻoi loa i loko o ka iapaau ana o ka panic kāna hana, a obsessive-compulsive kāna hana.
Nānā akula au i ka leo i ka medicament i ka loa haʻahaʻaʻo Solomona no α2-, α1- a me ka β-adrenoreceptors like hoʻi me ka m-holinoretseptorami, dopamine, 5HT1-me, 5HT2-e like me ka histamine H1-receptors.
Hana psychomotor oihana aʻe o ka lāʻau "Paroxetine"? Reviews o nā kauka e olelo aku i ka lapaau i ole ia ma luna o ke kanaka psyche negatively. Eia hoʻi, ka mea, 'aʻole i potentiate i ka depressant hopena o ka ethanol ma psychomotor hana.
Allegedly noiʻi i hōʻike 'ka antidepressant ua nawaliwali ho'ā' ia ka waiwai wale ina mea ua lawelawe ma dosages ma luna ma mua o ka poe i koi 'ia no ka inhibition o serotonin reuptake. Mākou hiki ole ke olelo i keia k 'aʻole ole i ka nui loli i loko o ke koko, pae, EEG a me ka naau kōmi.
Nā pharmacokinetics o ka 'inikua mea
lāʻau "Paroxetine" e like me ke kemu? Na Ke Kumu no ka hoʻohana 'ana, maoli kauka e olelo aku nei ia ma hope o moʻolelo hooponopono ana o na hana waiwai ke kemu, mai ka digestive'āpana, a ua metabolized ma ke akepaʻa.
Na wahi lehulehu o ka medicament i loko o ke koko ma o kā 1-1.7 pule ma hope o he lālā o ka lāʻau lapaʻau. Kaʻeleu 'Oponopono o ka lāʻau ua nui māhele i loko o nā'aʻaʻa. Ma keia hihia, ia mea ua loaʻa hoʻokahi wale pakeneka i loko o ka wai koko. Palapala a me na nā polokina o ka mea o 95%.
Antidepressant metabolized ma ke akepaʻa. E like me ka hopena, AEeOEXAaI metabolites i hana. Ka mea, koke eliminated mai ke kino, a i ka haʻahaʻa pharmacological hana, a i ole ia i ka pākōlea ole o ka lāʻau.
lāʻau "Paroxetine" like hōʻike? 'Ōlelo Aʻo, pharmacists lākiō i hoakaka ia ma kahi o 64% o kaʻeleu waiwai ua hookuu pu me ka mimi, oiai ka i koe, 36% - i loko o ka naʻau liʻiliʻi (ma ka bile).
Nā pharmacokinetics o ka lāʻau i loko o kūikawā lapaʻau wahi, i hiki
I ka lehulehu o kaʻeleu waiwai i loko o ke koko, wai koko kēia piʻina ma ka 'aʻe o ka hakuʻala a me akepaa, e like me ka mea kūpuna.
Nāʻikepili no ka hoʻohana ana i ka 'inikua mea
Ma kekahi hihia, e hoakaka nā mea maʻi antidepressant "Paroxetine"? ma ke noi o ka mea paahana alakai iloko ona i kakauia na kēia papa inoa o kāuʻikepili:
- i kekahiʻano o ke kaumaha, a me ka wi endogenous, kū'ē, a ua hele pu me ia e ka iini;
- panic kāna hana, a me agoraphobia;
- obsessive-compulsive kāna hana (OCD ole abbreviated);
- generalized uunu nui kāna hana;
- nohona uunu nui kāna hana, a no laila,-kapaia kaiapili phobia.
Contraindications i ka hoʻohana 'ana o ka' inikua mea
Ma kekahi mau hihia, i ole hihia hiki ole ke hoʻohana 'ia ma nā mea maʻi antidepressant "Paroxetine"? ma ke noi o ka mea paahana alakai ka loaʻa o ka kēia papa inoa o nā contraindications:
- lolelua ka epilepsy;
- concurrent ana o ka monoamine oxidase nā mea kūpale, e like me he mau-pule au ma hope o kā lākou withdrawal;
- na keiki o ka makahiki;
- gestation au;
- Hypersensitivity i ka lāʻau eiiiiiaiou;
- i breastfeeding.
E hoʻohana i me ka lōʻihi mālama nui
Ma ka hihia e e lāʻauʻai ana o antidepressant "Paroxetine"? Na Ke Kumu no ka hoʻohana hākālia nō i ua lawelawe iho la no keia makaukau me ka mālama nui i nā mea maʻi i ake e loaa, huina-panina glaucoma,ʻaʻa puʻuwai e hemahema, Mania, benign prostatic hyperplasia, convulsive Hawaii, cardiac kāna hana, epilepsy. Eia hou, i ka concurrent pono o ka helu kuhi ka lapaʻauʻia a me cardioversion, e like me lapaʻauʻia e hoomahuahua i ka pilikia o ke kahe ana ke koko. Mākou e uku mau noonoo a hiki i ke alo o ke kamepiula kumumea no ka kahe ana ke koko kāna hana, a mea conducive ia ia mai Hawaii.
Antidepressant "Paroxetine": pehea e lawe i ka laau?
Mākou e noʻonoʻo 'ana i ka lapaʻauʻia ua lawe hōʻike waha' koke i ka lā (i loko o ke kakahiaka) i ka aina kakahiaka. Papa e e ale a pau, holoi iho la me ka akaka ka wai.
Iloko o ka mea mua ekolu pule ma hope o ka hoʻomaka 'ana o ke lapaau i ka laʻau heluna ua like pākahi. Ua Ua a laila like (inā pono).
Ma hooloihi ae i kaumaha waiho dala o ka medicament He 20 mg koke i ka lā. Inā koi 'ia, i ka mahele lāʻau ua i nā hoomahuahua ia ka 10 mg. Max loaa i ka lāʻau e ole mamua o 50 mg.
No ka obsessive compulsive kāna hana loiloi mua mahele lāʻau o ka antidepressant He 20 mg no ka lā. Mahope, ka mea maoli he 10 mg. Ke paipai awelika kela la i keia mahele lāʻau no ia i haiahū kūmau o 40 mg. mea hiki e mahuahua i 60 mg Ma huʻi mea.
Inā ke hoʻomanawanui i ka panic kāna hana, e hiki initially lawe mai i ka 10 mg o ka lāʻau no ka lā. E emi i ka hiki pilikia o ka panic symptoms i loko o ka hope mahele lāʻau o ka lāʻau ua mahuahua ka 10 mg. Ma awelika, ka wā e like me ka haiahū kūmau mea maikaʻi nō ia i hoʻohana 40 mg "paroxetine" i loko o na hora, i ka i kā mākou helu - 50 mg.
I ka nohona phobia a nohona uunu nui kāna hana medicament loiloi mua ka leo e ole oi 20 mg no ka lā. Inā ma hope o ia i ka lapaau i ka makemake ia i ole, ua loaʻa, a laila, 2 pule ka mahele lāʻau ua kiʻekiʻe o mahuahua i ka i kā mākou, i mea mai ka 50 mg no ka lā.
Ma generalized ka iini kāna hana pākōlea, a me ka loiloi mua ka leo o ka medicament He 20 mg no ka lā
Inā diagnosed ka hoʻomanawanui me ka akepaʻa a me nā konāhua ka hoʻokō 'ole, ka paipai mahele lāʻau e e 20 mg no ka lā.
Mua kanaka i ka lā hiki ke hoʻopau i hou aku 40 mg o ka lapaʻauʻia.
I mea e pale aku withdrawal symptoms lawe i ka lāʻau 'ana ua pono ke kiʻekiʻe.
hihia o ka overdose
He nui na hihia o ka overdose me antidepressants e like me "Paroxetine", "Fluoxetine"? Mau loea, e hoailona oukou i ka mea maoli he kūlana maikaʻiʻole i ka hoʻohana 'ana o ka helu nui o nā huaale i ke kanaka kino. Ke hoʻomanawanui ka hoao ana nausea, maloo waha, sinus tachycardia, ka luaʻi, convulsions, tremor, bradycardia, mydriasis, manaʻo pīhoihoi, irritability, sweating, nystagmus, mahuahua ke koko, somnolence, a me nodal pāpana.
Ma 'ano pohihihi keia manawa oiai ka hoʻohana' ana i ka lāʻau a me nā psychotropic ai ', a me ka waiʻona i comatose ahonui, a me ka oko o ka PAaIEN ma ECG. I loa overdose, i ka hoʻomanawanui mea serotonin maʻi pale a me ka rhabdomyolysis.
He aha e hana i loko o ia mau wahi, i hiki? Ma ka hihia o ka lāʻau overdose "Paroxetine" E e gastric lavage, a lawe i ka ho'ā 'kalapona. Inā pono, symptomatic lapaau.
ʻaoʻao waiwai
He aha e hiki i "Paroxetine" kaʻaoʻao 'ole o ka lapaʻauʻia? Reviews o nā kauka e olelo aku i keia mea paahana maoli kōkua e hoʻomōhala adverse reactions. O nā ka ana ma lalo nei a me nā maʻi:
- Ma ka hapa o ka Central ko mākou hopohopo'ōnaehana a me kaʻike ākea ko mākou hopohopo'ōnaehana: Mania, drowsiness, ka hilahila, tremor, serotonin maʻi pale, luhi, hallucinations, Kanikani'āʻula, nervousness, pōniuniu, depersonalization, luhi, panic ho'āhewa wale, ke kāʻili 'ana, manaʻo pīhoihoi, amnesia, extrapyramidal kāna hana, myoclonus, uunu nui.
- Musculoskeletal'ōnaehana: Muscle nawaliwali, arthralgia, myopathy a me myalgia.
- Makaukau: blurred a blurred hihiʻo me ka a pau.
- Urinary'ōnaehana: pinepine urination a urinary ka mālama.
- Digestive'āpana: mahuahua ai ua hoʻemi ikaika loa ka makemake, hepatitis, ono loli, maloo waha, nausea, diarrhea, ka luaʻi, a me ka constipation.
- Reproductive'ōnaehana: anorgasmia, moe dysfunction, hyperprolactinemia a galactorrhea, impotence a me ka ejaculation kāna hana.
- Mea'ōnaehana mānowai koko'ōnaehana: orthostatic hypotension.
- Allergy: ka ohane, poʻe noʻonoʻoʻole, angioedema, a me ka urticaria, ecchymosis.
- Other likeʻole: rhinitis, sweating, kūpono 'secretion o antidiuretic hōmona, hyponatremia.
AaOIeIOUIeXAOAaIN a me nā 'inikua ano
Ke i ka wā hoʻokahi 'ana o nā antacids aʻole e pili mai ka pharmacokinetic kiko'î a me ke omo o ka lāʻau "Paroxetine".
Contraindicated no ka hoʻokahi-manawa hoʻohana ana i ke dala me ka Mao nā mea kūpale mua mākou.
I ka wā hoʻokahi? Eaia medicament "paroxetine" me ka ai 'i inhibit ake nā'ūhū, pono ka hookuu ana o ka mahele lāʻau mua.
Antidepressant hooloihiia kahe ana ke koko ma luna o ke kāʻei kua o kekahi-manawa i "o ka warfarin."
I ka wā hoʻokahi 'ana o ka medicament "paroxetine" me tricyclic antidepressants, aspirin, atypical neuroleptics, NSAIDs, a' o ia hoʻi phenothiazine papahana paipai 'ana i ke koko clotting kaʻina.
I ka wā hoʻokahi hoʻoponopono me ka serotonergic konohiki (e like me "tramadol" a me ka "sumatriptan") hiki wale alakai i ka hoʻokāʻoi 'serotonergic ole.
He nui ke hoomanao!
E pale i ka hooulu ana o ka neuroleptic maʻi pale (malignant), he lāʻau me ka lōʻihi mālama nui "Paroxetine" i hoakaka ia i ka hoʻomanawanuiʻana, ka poe i lawe antipsychotics.
Mua kanaka ma luna o ke kāʻei kua o ka lāʻau i hoʻomōhala hyponatremia.
I ka na hoailona mua o ke kāʻili 'ana a me ka Mania antidepressant Inc ua hoʻi i kāpiliʻia.
Iloko o ka mua pule o ka iapaau ana me "paroxetine" pono akahele ka mālamaʻana o ka hoʻomanawanui ma muli o ka hiki he pepehi anaʻia iā iho.
Ma Inc E hookaaokoa i ka io kanakaʻona mau nā mea inu aie i kā lākou hoʻokāʻoiʻawahia hopena.
Pediatric hoʻohana
Uluwehi O "Paroxetine" ua i hoakaka i na keiki, e like me kona ola a me ka hopenaʻoi loa i loko o ka iapaau ana o nā mea maʻi i loko o keia pae i ole, ua hoʻokūpaʻa.
Antidepressant "Paroxetine": counterparts
Ka lāʻau 'hiki auou caiaiai e "Paroxetine"? It E e kaulana i keia ka lapaʻauʻia, loaʻa nō loa he mau counterparts. Iwaena o lakou, ka mea makemake e kupono e kahińuli i ke kēia mau ai ': "Reksetin", "Adepress", "Pliz", "Apo-Paroxetine", "Aktaparoksetin", "Paxil", "sertraline", paroxetine hydrochloride hemihydrate, "" Sirestill "a no laila, ma luna o.
E kuai a pau o kēia mau lapaʻauʻia ma ka hale kūʻai lāʻau lapaʻau, e hiki wale ma kuhikuhi.
Reviews o medicament
Uluwehi O "Paroxetine" i kekahi wahi lihi iki o ka poʻe'ē he hōʻike manaʻo, nā mai ka 'Oihana a me nā mea maʻi mai. Ma ka kekahi lima, ka mea, ua hoonani aku la ia no ka mea ka mea, ka poʻea pau i ka kokololio hoʻopau ana i kekahi 'ano o ke kaumaha (a me ka wi endogenous, kū'ē, a ua hele pu me ia e ka iini), e like me ka pono me panic, obsessive-compulsive, generalized a me ka pilina-ka iini kāna hana. Ma ka 'ē aʻe - he nui loa nā mea maʻi e olelo aku nei ia mahope koke iho o ka lāʻau e hoʻomōhala loa i ka nui helu o adverse reactions. E like me ka hopena, kanaka i hiki i ke hooki i ka iapaau ana.
I mau, mau loea, e hoailona oukou i ka "Paroxetine" - keia mea he loa pono a me ka efficient lāʻau Makuakane me ka hana häʻawi mai ai iä ia. Naʻe, ka mea hiki ke hoʻohana wale no kona Manao iho la ia mea hoʻomalu.
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