Ola kino, Hoomakaukau
Loperamide hydrochloride. Loperamide hydrochloride - manual
He aha mea i ka lāʻau "Loperamide hydrochloride '? A hulina pane i keia ninau hiki ke loaʻa i loko o ka mea i hoakaka ia ma ka 'atikala. Eia hou, e hai aku mākou iāʻoukou i loko o au mamuli e pili ana pehea e lawe i ka ka lapaʻauʻia, ka wā a ma ka laʻau heluna.
kekahi mau 'ike
Ka medicament "Loperamide hydrochloride" mea he symptomatic lāʻau i ua pinepine hoʻohana i ka hana huʻi a me ka maʻi diarrhea. Kēia lāʻau 'ua kuaiia me ke kuhikuhi, a kuai lilo aku la i kaʻaneʻane na hale kūʻai lāʻau lapaʻau ma ka affordable kumukuai.
Pharmacological 'ole
E hoomakaukau ai "Loperamide hydrochloride" aʻo i ua punana ma ka carton, ho'ēmi i kā motility a me ka leo o ka laumania Muscle o ka naʻau liʻiliʻi, a inhibits peristalsis o ke kino, nui mahuahua ka maalo manawa o kona Contents. Ke'ī mai, ka mea a hooku iho la medicament ka lawe antidiarrhoeal hopena. It E e hoʻomaopopo i ka lāʻau "Loperamide hydrochloride" hoʻomaka i ka hana nui koke. I? Eaia o keia k i loko o ka pākōlea ia mau no e pili ana i 4-6 hola.
Pharmacokinetics
Oia ka medicament ka paka i loko o ka naʻau liʻiliʻi mea he ilihune (ma kahi o 40%). Aie i ka mea kiʻekiʻe similarity i receptors o ka intestinal pā, e like me keʻano kiʻekiʻe o biotransformation i ka hooholo mua ma ke akepaʻa wai koko pae o unmodified ke keʻena ma hope o ka loaa ana i na mea 2 mg (1 mea hōʻikeʻikeʻuʻuku) ka emi o 2 ng / ml. ʻO kā mākou lehulehu o ka hana waiwai ma hope o hoʻohana pāʻoihana ua hiki aku ma hope o ma kahi o 2,5 hora, a ma hope o nā capsules - ma hope o 5 hola. Paa i ka wai koko nā polokina ia lŘlŘ i loko o 97%. Kēia lāʻau ua metabolized i loko o ke ake, a ua loko ma ka hapa mai o ka mimi, like conjugates me ka bile, e like me me ka feces.
Release palapala o ka lapaʻauʻia a me kona haku mele 'ana
E hoomakaukau ai "Loperamide hydrochloride," i ka hoʻohana 'ana o i ua hōʻike i hoakaka ia, ua-market i loko o ka palapala:
- Waiwai ka pauka no ka pāʻoihana.
- 2 mg na papa, e hoonoho iho i loko o ka carton 50, 30, 20 a me 10 apana.
- 2 mg capsules waiho i loko o ka AEeAaOA 30, 20 a me 10 apana.
- Gelatin paakiki capsules yellow, i pihaʻi me he keʻokeʻo ka pauka me kaʻeleu ke keʻena - loperamide hydrochloride. Kēlā me kēia mea hōʻikeʻikeʻuʻuku he 2 mg oʻeleu waiwai. Ma waho poe medicament kekahi i loko o kona haku mele 'ana, a kākoʻo nā mea hoʻohui: talc, ke kulina pia, lactose, makanekiuma stearate a me colloidal ka silica i. Gelatin capsules i nā pāʻoihana i loaʻa i loko o ka carton 20 a 10 apana.
Where'ē aʻe no ka hana 'Oponopono loperamide hydrochloride? I ka hana ana o keia waiwai ma ka pharmacology a leie aku ai 'e like me "Imodium" a me ka "Diara". Eia naʻe, kona pakeneka i loko o kēia mau mea haʻilula keimikala mea nui uuku ma mua i loko o ka hoʻoili medicament.
Uluwehi O "Loperamide hydrochloride": ka mea i manaoia?
E like me na kuhikuhi, ka lāʻau ua koi 'ia e lawe i ka i kēia hihia.
- E normalize i ka noho ma ileostomy.
- I ka metabolic kāna hana, a intestinal omo, a i ke kumu e koke, a drastic loli ma kaʻai a me ka mau haku mele 'ana o kaʻai (no ka laʻana, ma kaʻai, ma luna o ka hele ana).
- Me he kākoʻo lāʻau i loko o infectious diarrhea.
- Like symptomatic lapaʻau no ka huʻi paha maʻi diarrhea (allergic, pāhawewe, lāʻau a mea naʻau me Kinohi).
Contraindications i ka hoʻohana 'ana o ka lapaʻauʻia
Ma kekahi mau hihia, e hiki ole hoʻohana i ka lāʻau "loperamide" (papa)? Na Ke Kumu haawiia ka lapaʻauʻia Hawaii i ka mea i pono no:
- intestinal iaʻi;
- diarrhea, a i kaua kipi ma muli o ka hī koko, huʻi pseudomembranous enterocolitis 'ole' ē aʻe nā mea palahēhē o ka digestive'āpana;
- diverticulosis;
- huʻi ulcerative colitis;
- hypersensitivity.
Ua E hoi e kaulana ia mau antidiarrheal ai 'ia nā keiki e e hoakaka ia wale i 4-makahiki. Eia hou, e like me na kauoha, 'o ia hoʻi "loperamide" ua contraindicated i loko o ka trimester mua o ka hāpai keiki, a i lactation. Me ka malama nui i ka lāʻau 'ua hoakaka ia no ka ake ole.
Ka medicament "Loperamide hydrochloride": kauoha no ka hoʻohana
Papa a me capsules o ka lāʻau, e e lawe hōʻike waha me Kamehameha a mama. Ke laʻau heluna o ka lāʻau hilinaʻi nui ma luna o ka makahiki o ke ahonui a me ka maʻi oolea.
Ma huʻi diarrhea i loko o nā mākua e like me ka mahele lāʻau mua lawelawe 4 mg o ka lāʻau, a laila, - e 2 mg ma hope o kēlā me kēia defecation (ina ke noho nei nō wai).
I ka maʻi diarrhea mua mahele lāʻau o 2 mg. Hope Inc no nā mākua e e? Ieoaeunoai ai i ua 1 a me 2 manawa no ka lā o ka hoʻomanawanui i ka noho alapine (frequency). ʻO kā mākou kela la i keia mahele lāʻau - 16 mg.
Ka pākōlea hopena o ka lawe ia ka lāʻau e hoʻomōhala ana i loko o 48 hola. Inā, nae, no ka 2-4 lā, ka hoʻohana 'ana i ka 16 mg o ka lāʻau kēlā lā, e hiki ole kū i ka makemake hopena, oe e mau nīnau aku i ke kauka, ka mea i ho'ōla aʻe iā lākou, e noonoo i kaʻike,. E ho ohana ana i ka lāʻau 'hiki e hou, akā, wale nō inā' ilepili lapaʻau a eaioiuo 'aʻole i normalize i ka noho.
Like no na keiki, e like me ka lāʻau e hoʻohana wale 4 makahiki. Ka mahele lāʻau Ua hoi e kaukaʻi ma ka makahiki o ka hoʻomanawanui, a me ka oolea o ka maʻi.
Na kamalii uuku mai ka 4 a hiki i 7 makahiki, pono e haawiia ka lāʻau 3-4 manawa i ka lā a hiki i 1 mg. Duration o ka Inc mea 3 lā. Children mai 7 a hiki i 12 makahiki lawelawe eha manawa i ka lā 1 papa no 5 mau lā. I ka huʻi diarrhea loiloi mua laʻau heluna keiki e e 1 mea hōʻikeʻikeʻuʻuku. ʻO kā mākou kela la i keia mahele lāʻau no nā keiki - 8 mg.
Inā he keiki ua diarrhea malama ma hope o kēlā me kēia hana o ka defecation i loko o ka lōʻihi manawa, o kela mea keia manawa ia e haawiia mai e 1 mea hōʻikeʻikeʻuʻuku, akā,ʻaʻole oi aku mamua o 6 mg no 20 kg o ke kino ke kaupaonaʻana no ka lā. Inā ke kamaiki, aole ia e hele i ka 'Ia oi ma mua o 12 hora, a ma hope o normalization o ka noho? Eaia imua o ma ka lāʻau i ka manao e hooki aku.
lāʻau overdose
I Ina o ka overdose me keia k i loko o ka hoomanawanui kēia mau deviations hiki ke malama.
- haunaele ma ka ōhumu o ka neʻe 'ana;
- constriction o na haumana;
- nanea ana;
- drowsiness;
- hoomahuahua ae la lakou skeletal Muscle leo;
- na naau oʻu iaʻi;
- naehana hanu kaumaha.
E hana i na pathological Hawaii kauka pinepine lāʻau "Naloxone" ua hoʻohana 'ia me ka i ka wā hoʻokahi symptomatic Inc.
ʻaoʻao waiwai
It E e kaulana ia ma hope o ke noi ana o ka la hoomalolo "Loperamide hydrochloride" nā mea maʻi e 'ike kekahiʻaoʻao ona. Loa pinepine ka mea ana me ka hooloihi ae i hoʻohana o ka lāʻau. Pela poe medicament hiki i ke kēiaʻaoʻao ole:
- flatulence;
- electrolyte abnormalities;
- ka luaʻi;
- intestinal cramps;
- pōniuniu;
- gastralgia;
- nausea;
- hypovolemia;
- drowsiness;
- maloo waha.
I na keiki opiopio, he lāʻau pinepine ke kumu discomfort i loko o ka abdomen, like hoʻi me ili rashes. Loa kākaʻikahi medicament "Loperamide hydrochloride" e hoʻonui i ka urinary ka mālama 'ole intestinal iaʻi.
Inā ma hope o 2 lā i kēia mauʻike manaʻo mai i nalo, a me ka hoʻomanawanui, aole ia i haha aku maikaʻi, oe e mau nīnau aku i ke kauka, nana no e hoonoho i ka mea'ē aʻe (like) huahana. Inā he lāʻau,ʻaʻole i kōkua, ia mea maikai, e nānā i nā mea palahēhē mea i diarrhea.
lāʻau hana kūleʻa
E like me na kuhikuhi, oiai ka noi o hoʻomākaukau "Loperamide hydrochloride" a me ka "Cholestyramine" mua ka hoʻokōʻana e emi iho. Inā 'oe pono e hoʻohana' ana i ka lāʻau a me nāʻano "Li-trimoxazole" a me "Ritonavir", alaila oe e ike i kona bioavailability ua me ka nui loa mahuahua.
Cautions
Uluwehi O "Loperamide hydrochloride" E e ia me ka lōʻihi mālama nui i loko o hepatic hoʻopilikia. Ua ua no hoi e waiho i ka hana ia i loko o kēia mau wahi, i hiki lapaʻau kahi inhibition o intestinal peristalsis. I ka wa e kaawale aku o ka pono pākōlea kanawai ma hope o 2 lā ma hope hooponopono ana o ka lāʻau ia mea kupono, e hoomaemae i kaʻike, o ke kauka, a hoʻopau infectious Kin diarrhea.
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