Ola kino, Hoomakaukau
"Oseltamivir": aʻo no ka hoʻohana 'ana, analogs, he hōʻike o ka lāʻau
No ke aha la i koi 'ia ka lāʻau "Oseltamivir"? e ho'ākāka 'ia ma ka iki ae aʻo no ka hoʻohana' ana, analogs, nāʻikepili a me contraindications o ka lāʻau, e. E hai mai no hoi oe e pili ana i ke ano o ka mea au e kūʻai mai la medicament, He aha ka waiwai ka mea, ua loaa, ina paha ma kaʻaoʻao ona, a no laila, ma luna o. D.
Ke kinona, 'ole, hōʻikeʻano o ka lāʻau
Ma ke kuai ana o ka lāʻau hele mai i loko o ka palapala o ka melemele-keʻokeʻo capsules. "Oseltamivir" - He He prodrug. I ka kino, ka mea, ua hydrolyzed a ua hoohuliia mai i ka hana 'Oponopono - oseltamivir carboxylate.
Ma waho aʻeo ia na capsules, a me ka medicament ua hookuu ia ma ke ano o ka malamalama he lepo no ku una mai paha.
hiʻona ka lapaʻauʻia
lāʻau "Oseltamivir" Pehea 'aʻole ia hana? Na Ke Kumu ma ka noi hākālia nō i ka pākōlea kanawai o keia ka lapaʻauʻia ua nānā 'ana i suppression o ka hana o nā'ūhū, a i aia ma ka ili o ka virion maʻi palū mea hoʻomaʻi.
Ma ka loaʻa 'ana o ka medicament i loko o ke kanaka kino kona papa kuhikuhiE ke keʻena ia iho me ia i kaʻeleu metabolite. Penei, oseltamivir carboxylate selectively inhibits neuraminidase. E like me ka hopena o ia waiū pohaku mea hoʻomaʻi aeea multiplication kaʻina.
E like me ke akamai, e lawe i kēia ka lapaʻauʻia ai e haawiia mai i loko o 35 hola ma hope o ka hoailona mua o ka maʻi palū. Wale ma keia ala hiki ke hoemi i ka lōʻihi like 'ole o ka maʻi ma 30%, a me ka pahiki o complications a me ka oolea o symptoms - 40%.
Pharmacokinetics o ka lāʻau
Paha ka lapaʻauʻia ka paka "Oseltamivir"? Na Ke Kumu no ka hoʻohana i ka 'ia ma kahi o 90% o ka oseltamivir posapahate ke kemu i loko o ka gastro-intestinal'āpana. Kaʻeleu waiwai ua hoohuliia i ka carboxylate o oseltamivir, a laila, komo i ka systemic holo.
About 3% o ka hana 'Oponopono ua paa ia i ka wai koko nā polokina. Kona bioavailability mea o ka hola 76-85% a me ka hoʻopau hapa-ola - 120 minuke.
Mai kanaka oseltamivir carboxylate ua loko ma nā puʻupaʻa (ka hola 80%), a gut (20%). Hapa-ola o ka lāʻau mea 6-10 hola.
nāʻikepili
No ke aha la i koi 'ia ka lāʻau "Oseltamivir" (aina pūʻulu -. Antiviral Luna)? E like me na kuhikuhi, ka medicament ua hoʻohana 'ia no ka hana maʻi palū A a me B. kekahi, ka mea, ua pinepine ia no ka Kāohiʻana o ka mea hoʻomaʻi ka maʻi.
Contraindications
Anei contra "Oseltamivir" (hōʻike o ka la hoomalolo, ua hōʻike mai iā ia ma luna)? E like me na kuhikuhi, ka lāʻau ana ua pāpā ma:
- Hypersensitivity i ka hana 'Oponopono;
- ʻaʻa puʻuwai 'ole (palekana a me ka hopenaʻoi loa o ka lāʻau i loko o kēia nā mea maʻi i ole, ua hōʻike');
- i na keiki kaikaina ma mua o 1 makahiki (he mea maopopo like ai i ke kahua o ka BBB i loko o nā keiki);
- hāpai keiki, a breastfeeding (ka mea, ua hoʻi i hōʻikeʻia ka lāʻau ua excreted ma ka umauma i ka waiū o nā wāhine, a me ka mea ia e loli ai i ka fetus).
Ua E hoi e kaulana i keia ka lapaʻauʻia ua i paipai no na keiki ma lalo o 13 makahiki, e like me ka poe akamai i ole, ua manao palekana a me ka hopenaʻoi loa o ka 'Oseltamivir' no ka Kāohiʻana a me ka hana o ka maʻi palū.
Uluwehi O "Oseltamivir": kauoha no ka hoʻohana
Vidal (laau Akanahe) he hulina 'ike ma luna ana, a ma ka laʻau heluna oe e lawe i ka lāʻau ma ka nīnau. Naʻe, ka mea e e hoʻomaopopo i koi 'ia ka lāʻau e wale kauka. Ma hope o nā mea a pau, wale i ka hoao ana i ka hoʻomalu e e hiki ke koho i ka akau lapaʻau regimen, i koke a me ka pono hoʻopau i kaʻawaʻawa loa symptoms o ka mea hoʻomaʻi maʻi.
No laila, i loko o ka laʻau heluna ua hoakaka ia "Oseltamivir"? Na Ke Kumu no ka hana hōʻike 'ana i keia k E e hoʻohana i loko o 2 lā ma hope o ka hoouka kaua ana o ka hoailona mua o ka maʻi palū.
Children mua ma mua o 13 makahiki a me nā mākua me ka lāʻau lawelawe i loko o ka nui o ka 75 mg palua i ka lā i 5 mau lā. It e e koke kaulana ia e hoʻoulu ai i ka laʻau heluna o ka lāʻau (e laʻa me, i i 150 mg no ka lā) i i alakai i ka māhuahua pākōlea hopena.
Inā 'o ka lāʻau' oe makemake i ka hāʻawi aku i nā keiki elemakule 1-12 makahiki, ka laʻau heluna ua like ke kaumaha ma muli o ka keiki ka kino ke kaumaha.
E pale maʻi palū i nā mākua a me nā keiki ma luna o ka 13 makahiki i hoakaka ia 75 mg 1 kekahi manawa mamua no ka 6 pule ma ka lā (e like, i ka maʻi laha).
Hoʻomanawanui iki mai me Cl creatinine emi o 30 ml no minuke koi? Iaea laʻau heluna (75 mg hookahi no 5 mau lā o ka lā).
ʻaoʻao 'ole o ka lāʻau ma hope, inu
Kekahi adverse reactions i hoʻomaka ai ma hope o aaieieno? O 'Oseltamivir' hoomalolo? Na Ke Kumu ma ke noi mai nei i ka loa mau hoike adverse reactions i ka nausea a me ka luaʻi. Ma ka hapanui o na, mau 'ole e mehana ai moderately i olelo ia, a hookuu ana i loko o nā lā mua o ka nohoʻana.
Ua E hoi e kaulana ia i loko o kekahi nā mea maʻi, i nā mea maʻi e loaa ana i ka lāʻau ma lalo o ka nāʻanaʻana, hoʻomōhala bronchitis, vertigo, Kanikani'āʻula, lolelua ka angina, pseudomembranous colitis, anaemia, pneumonia, fractured humerus, peritonsillar abscess a me ka mai kuni.
Loa pohihihi keia i ka lawe ana i ka lāʻau "Oseltamivir" kanaka, he mau abdominal eha, kōkua lohe, nosebleeds a me conjunctivitis. Ma ka hapanui o na, mau reactions ana wale i kekahi manawa, a ua nalo ma luna o lākou iho, mamua o ka neʻeʻana Inc. Oiaʻike manaʻo mai i koi discontinuation o ka lapaʻauʻia.
Ma hope mai o ka manawa i oleloia ai o antiviral lāʻau i loko o nā keiki a me nā adolescents i akaka ia adverse loa. Mau nā i keia mau mea e like me ka poʻe noʻonoʻoʻole, ʻawahia epidermal necrolysis, haanou ana o ka olelo a me ka maka, arrhythmia, ka hilahila, ke kāʻili 'ana a me ka worsening o mimikō pele.
lāʻau hana kūleʻa
Ike i loaa i loko o ka papa o ka pharmacokinetic a me ka pharmacological haʻawina hoakaka ana o ka ulu o clinically nui lāʻau hana kūleʻa i keia k mea olelo lealea.
Na olelo hookomoia me ka lāʻau, ka mea, ua olelo mai ia i ka i ka wā hoʻokahi noi o ka medicament me ka probenecid hiki aku ai i ka mahuahua ma AUC o kaʻeleu metabolite o 2 manawa. Eia naʻe, mahele lāʻau hoʻoponopono 'aʻole koi' ia.
hihia o ka overdose
He aha e na symptoms ike i loko o nā mea maʻi me ka "Oseltamivir" nā māhele kiekie o ka waiʻona? Reviews a me nā kuhikuhi hoakaka ana i ka la i keia mau hihia ae la. Eia naʻe, hookahi dosages o antiviral lapaʻauʻia hiki i ka luaʻi paha nausea.
E hoʻonā i kēia mau symptoms, symptomatic Inc.
I Kekahi Mau koi no ka loaa ana ka lapaʻauʻia
He aha kou pono e ike i ka hoomanawanui, ma mua ka lawe "Oseltamivir"? Na Ke Kumu no ka hoʻohana (no nā keiki a me nā mākua e 'ike kekahiʻaoʻao' ole) ia Hōʻike i ka lāʻau mea i pili no ka makahiki vaccination. He i i hiki ole i ka hooulu ana o ka complications i ke hana i ka mea hoʻomaʻi maʻi, e like me nā mea palahēhē mea koʻohune.
Analogs medicament
"Oseltamivir" - he lāʻau i ua manao ia no ka lapaau a me ka Kāohiʻana o ka maʻi palū. He he antiviral Agena i pili i nā mea kūpale o neuraminidase. Kēia lāʻau ua olelo ike ma lalo o ka hao ka inoa "Tamiflu". Mall analogs ka mea, aole i nei. Ka hoʻopuniʻana, akā, kānaka wahi emi mahope hana, na kēia mau ai 'i pani ai, "Relenza", "Arbidol", "Flustol", "Kagocel" a me na mea e ae.
Reviews a me ke kālailaiʻana i ka laulā o ka lāʻau
E like me ka hoao hualoaʻa, a i loaa i loko o kaʻAmelika Hui Pūʻia a me Mexico, me ka hou nā mea hoʻomaʻi i ikepili koʻikoʻi i neuraminidase nā mea kūpale ( "Zanamivir" a me ka "Oseltamivir"), akā, ka mea e hoʻopale ai i ka mea 'ē aʻe pūʻulu - adamantanes ( "rimantadine", "Amantadine") .
Ua E hoi e hoʻomaopopo i ka poe akamai i ole i ka hopenaʻoi loa o keia k ma ka iapaau ana o ka maʻi palū Ua hoʻouka kekahi ma poʻe me ka maʻi puʻuwai a me ka ÷ naehana hanu maʻi.
E like me na kumu, ka lāʻau ho'ēmi i kā ka lōʻihi like 'ole o ka symptoms ma 1 lā, akā, i kēia mea wale nō i ka hihia ina ka iapaau ana i hope o hui' ana me ka hoʻomanawanui hoʻomaka 'ana i loko o ka mua mau hola.
I ka lā,ʻaʻohe ike loea 'ike ma luna paha o ka hopena o kaʻai ana o ka lāʻau ma luna o ka mea hiki wale mai o complications o ka mea hoʻomaʻi a infectious maʻi.
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