Ola kinoHoomakaukau

Ka lāʻau "Akineton": aʻo no ka hoʻohana 'ana, hōʻikeʻano, hōʻike manaʻo

Kaʻeleu waiwai "Akinetona" Ua biperiden hydrochloride. Papa lawa 2 mg oʻeleu waiwai. Eia kekahi, i ke alo o nā eiiiiiaiou (kulina pia, uala pia, lactose monohydrate, makanekiuma stearate, microcrystalline kelulose, copovidone, kalipuna hydrogen posapahate dihydrate, talc, maemae ka wai) kuhi i ka lāʻau "Akineton".

Na Ke Kumu no ka hoʻohana, ka Hawaii photo paipai i ka papa palapala o ka lāʻau i kokoke keʻokeʻoʻeleʻele, Valium palapala. Ma kekahiʻaoʻao o ka papa, aia o ka pilikia o ka beveled kea shape.

1 ml o ka pāʻoihana he biperiden lactate i loko o ka nui o ka 5 milligrams. Additional eiiiiiaiou i: injecting ka wai a me ka paʻakai lactate.

Pharmacological 'ole

Main 'Oponopono biperiden - holinoblokator kikowaena hana.

Ka hopena komo ai e kaumaha ana i ka hiki i ka cholinergic neuronal haʻawina i loko o ka striatum, i mea ka mall pa alima o ka extrapyramidal nenoaiu.

I ka lāʻau a nā ganglioblokiruyuschimi hookoia, antispasmodic a me ka lōpū oolea ka m-anticholinergic 'ole ma o ka periphery (antispasmodic).

E ho ohana ana i ka lāʻau 'kōkua hoʻopau lala tremor, i kupu ana ma ka hoʻohana o cholinergic ai' (e laʻa me, pilocarpine) a me ka catalepsy a me ka Muscle rigidity i loko o nā mea maʻi loaa neuroleptics. Ka mea, i ka hiki e induce manaʻo pīhoihoi.

Pharmacokinetics

"Akineton" e paa ana i ka wai koko nā polokina ma 91-94%. Wai kokoʻae e e 11,6 ± 0,8 ml / min / kg kino ke kaumaha. A hookahi mahele lāʻau o ka moʻolelo no ka hoʻomanaʻo i ka bioavailability o ma kahi o 33 ± 5%.

Hele i loko o ka umauma o ka waiu.

Biperiden maopopo metabolized i loko o ke kanaka kino. I mimi, i ka waiwai ua i nānā 'ia ma unaltered palapala. Ka nui metabolites i bicycloheptane a me ka piperidine, i mea auoiaea, mai na feces a me ka mimi.

Elliminatsiya lawe mai i loko o nā kūlana, a me ka hapalua o ke ola (T 1/2) o 90 minuke i ka pae mua a me ka 24 hola - i ka lua o ka pae. I ka poʻeʻelemākule nā mea maʻi, me ka hapa-ola ke mahuahua kūpono kou.

nāʻikepili

"Akineton" hoʻohana 'ia i loko o extrapyramidal kāna hana e poloʻai pule ma ka hooponopono ana i kekahi mau lapaʻauʻia (neuroleptics, antipsychotics).

Nō hoʻi, i ka lāʻau ua hōʻike no kaʻike, o ka maʻi Parkinson ka maʻi pale, parkinsonism (hope paha lawelawe ma ka hui pu ana, Inc me ke kumu)

Contraindications

Ua i hōʻike 'ia ke kumu o keia k ia oe e hypersensitive i ka hana' Oponopono o ka lāʻau "Akineton".

Na Ke Kumu no ka hoʻohana hoʻomaopopo 'o ia i ka lāʻau e e käpae' ia ma kaʻike, o ka maʻi i loko o ka hoomanawanui e like me prostate hoʻonui, huina-panina glaucoma, obstructive hou i loko o ka naʻau liʻiliʻi (pylorus stenosis, lolo ileus Kin).

Arrhythmia, epilepsy, umauma, e ai ana, kūpuna, hāpai keiki nō nā kumumea i loko o i "Akineton" lawelawe me ka mālama nui.

ʻaoʻao waiwai

CNSʻaoʻao waiwai i hoikeia asthenia, luhi, lethargy, nawaliwali, numbness, pōniuniu, manao o ka mea e hopohopo nei, uunu nui, iaiyoe hoʻopilikia, ka hilahila, hallucinations, catalepsy, lāʻau kaukaʻi lāʻau "Akineton".

Na Ke Kumu no ka hoʻohana kamailio anaʻaoʻao-mau waiwai, a me ka hapa o ka hihio - mydriasis, mai ka pioloke o ka noho.

Cardio-vascular'ōnaehana ua wehewehe aku e kaoo ana o ka naau i kela (tachycardia); kekahi manawa, - deceleration (bradycardia); ka wā ana i ka pahu kui palapala o ka la hoomalolo - emi i loko o ke koko, (hypotension).

Ma ka hapa o ka digestive'ōnaehana - maloo waha, dyspeptic symptoms, constipation.

Ma ka hapa o ka pūnao - emi sweating.

Ma ka hapa o ka urinary'ōnaehana - i loko o nā mea maʻi me ka hoʻonui (hypertrophy) o ka prostate gland - hiki pilikia mimi.

Allergic reactions: wawe ma luna o kaʻili, maneo.

Nā Papahana O Ka E ho ohana i

No ka intramuscular, intravenous, a me ka haʻi waha papa palapala aole ia e pono e hoʻomākaukau ai "Akineton".

Na Ke Kumu no ka hoʻohana paipai ia Inc "Akinetonom" ano laulā, hoomaka mai ka meaʻuʻuku nā māhele, o ka mahele lāʻau oi iiyoaiiay, piʻi pū ke kaumaha ma muli o ka makemake pākōlea keia, a no kaʻaoʻao 'ole.

Nā mākua ma ka hoʻohana 'ana o ka una ka palapala o ka la hoomalolo hoʻomaka lapaʻau ma ka mahele lāʻau o ka 1 mg 1-2? Eaia i ka lā a me 2 mg māheleʻia i loko o nā nā māhele o ka lā. Eia, hiki e mahuahua ai ka laʻau heluna i 8 mg elua i eha puʻunaue nā māhele. Eia naʻe, mahele lāʻau e ole hoʻonui oi ma mua o 2 mg no ka lā. Mai oi aku ka mea i kā mākou laʻau heluna o ia hoʻi, 6 i TH-16 mg i elima mau lā. Single mahele lāʻau injectable lāʻau palapala e ole oi 2.5-5 mg. Kēia mahele lāʻau paha e hai hou ma hope o ka hapalua o ka hora, akā, i ka helu o ka papa hoʻomalu no ka lā e ole mamua o 4 manawa. ʻO kā mākou mahele lāʻau o ka medicament ma injectable palapala o 20 mg i elima mau lā. A hiki aku ka mea e pono ai ke mahele lāʻau ua hiki, alaila, he hoʻololi i ka? Eaia "Akinetona retard."

Akā, mai poina e pili ana i ke kanaka kokoke i kēlā me kēia hoomanawanui i loko o ka manawa i oleloia ai biperidenom Inc.

Extrapyramidal pathology i kupu mai ma muli o ka 'ai, inu ana i kekahi mau lapaʻauʻia (antipsychotics ole neuroleptics) pono paha o ka haawiia waiwai i loko o ka hookahi mahele lāʻau o ka 2 mg hōʻike waha paha parenterally. E hana hou i mau hoʻoponopono o ka olelo mai nā māhele i e kela hapalua hora. Eia naʻe, e like me ka hōʻike ma luna, ma ka helu o nā luna 'oihana e ole mamua o 4 manawa. Ka moʻolelo mahele lāʻau E e mahele ia i loko o kekahi i ekolu nā māhele.

Parkinson ka maʻi komo ai ka lawelawe ana i ka lāʻau 'hōʻike waha ma 6-8 mg ma 2-4 puunaueia nā māhele no ka lā, ka mahele lāʻau hiki ke i nā mahuahua mai ka 6-16 mg.

Children ma lalo o ka makahiki manao paipai i ka manawa kūpono o ka lāʻau i loko o ka injectable ano lohi, he hookahi mahele lāʻau o ka 1 mg a 0.2 ml. I ka makahiki, mai kekahi makahiki a hiki i na makahiki eono lawelawe 2 mg a 0,4 ml. Mai ka 6 i 10 makahiki - 3 mg a 0,6 ml. Kēia mahele lāʻau paha e hai hou ma hope o ka hapalua o ka hora me ka pilikia. Ma ke alo o adverse 'ole ma o ka hooponopono ana o ka lāʻau e e hele aku ka pahu kui.
Ma moʻolelo i ke ano o ka lāʻau Inc ma ka makahiki mai ka 3 a hiki i 15 makahiki o ka lawe i ka laʻau heluna o 1-2 mg i ka 1-3 hora i ka lā.

hiki ole i ka papa inu ma luna o ka nele opu, a me oe e inu i ka lōpū nui o ka wai. At hanana o undesirableʻaoʻao 'ole, mai ka digestive'ōnaehana e lawe i ka lāʻau' koke ma hope o kaʻai, hoemi i ka oolea o ke adverse hopena o ia hoʻi, "Akineton".

Na Ke Kumu no ka hoʻohana i ka 'ia i loko o ka hihia o ka nicotine i kaʻapu kōheoheo i loko o nā mākua maʻamau luna' Inc ua i lawelawe keia k, a me kona mahele lāʻau mea 5-TH-Tb-10 mg no injectable ano, akā, wale i ka hihia i olelo hooweliweli aku i ka hoʻomanawanui ka ola.

I kaʻapu kōheoheoʻana ke aloha phosphorus nā mea huihuina biperiden dosing ua lawe mai pākahi ke kaumaha ma muli o ka oolea o lesions. Omaka mai ka mahele lāʻau o ka 5 mg i loko o ka hihia o intravenous hooponopono, hai aaieieno? Hoʻomau a nalo kaʻapu kōheoheo i ka symptoms.

overdose

Overdose hoike mai ai ia haʻi anticholinergic 'ole ke kumu ma ka lapaau "Akineton".

Na Ke Kumu no ka hoʻohana 'ana, maoli kauka e lohe ai i ka mea i ka iapaau ana o keia kulana posimptomnaya (hoomau ana o ka mea'ōnaehana mānowai koko a me ka ÷ naehana hanu nenoai, oxygen Inc, hyperthermia? Iaea, he urinary catheter' ia paha, ina he pono). Pono ka hoike ana o ka cholinesterase inhibitor (physostigmine kuhikuhi) .

AaOIeIOUIeXAOAaIN

"Akineton" ana i ka hoʻohana 'ana i ka m-holinoblokatorami, ai' me ka antihistamine a me ka antiepileptic hana hoʻokāʻoi aʻe ana i olelo o ka hope. Eia naʻe, i ka wā hoʻokahi palapala noi o metoclopramide ho'ēmi i kā kona pākōlea ai. Aia definitive lāʻau incompatibility me ka ethanol. Ka hoʻokohu 'quinidine piʻina ma ka manawa o ka pilikia o ka ulu dyskinesia symptoms. ua hoʻokāʻoi 'M-cholinergic ai ka wā ana levodopa.

Pūnaewele a me ka kuai

E kūʻai i kēia k pono i ke kuhikuhi, e hoʻolako i ka pharmacist. E hoahu "Akinetona" Pono, e hooko me ka wela, 'ole. E. Ambient wela e ole oi aku mamua o 25 degere (Kelekia me ka unahiʻole). Mākou Pono i ka loaa ole o na keiki a hiki i ka hale "Akineton".

Manual haawi i ka holopapa ola o ka lāʻau - elima makahiki.

Cautions

Ka hoʻokohu 'ana biperiden i hāpai keiki, a breastfeeding (lactation) pono ikaika nāʻikepili.

Biperiden ke kiʻi i ka bebe ma ka umauma o ka waiu, e kauoha ana i ka? Aiaiiuie ole o breastfeeding i ka discontinuation o ka lāʻau "Akineton".

Product hōʻikeʻano o ka papa mai ia i loko o ka hoʻoholo 'ana ma o ka hookohu o ka biperiden i hāpai keiki, a lactation lawe i ka mooolelo o ka Loaʻaʻia kamepiula a hiki i ke keiki, fetus.

kekahi kamepiula ololi no ka iapaau ana me keia k kūpuna lilo. No laila, koho "Akineton" keia pae ana o kanaka me ka nui mālama nui.

Kickaha wa e kaawale aku o kekahi hoike o ka pono o ka mālama 'ia hoʻi i loko o kamaliʻi, o ke kumu i aole i pili i ka lāʻau' keiki "Akineton".

Description o ka la hoomalolo (manual) hoʻomōakaaka ka mea i ua koi mālama nui ia ka hoʻohana 'ana i kēia k i loko o nā mea maʻi me ka epilepsy paha fibrillation.

Me ka hooloihi ae i ana e hoʻomōhala lāʻau kaukaʻi.

Ka pilikia o ka withdrawal maʻi pale komo ai o ka holo cessation o Inc "Akinetonom".

i ke ano o ka waiʻona-i loaʻa nā mea inu e e käpae 'i ka Inc.

Iapaau ana me keia k pono ole ana, alaila, mai kipaku kaa a me nā haʻuki hana e noi mai ana kiʻekiʻe lehulehu a me ka kokololio psychomotor reactions, no ka mea, hāpai me ia i ka Loaʻaʻia pilikia ma muli o ai i ka pilikia o ka pōniuniu.

"Akineton". Na Ke Kumu no ka hoʻohana. analogs

Synonyms o ka hoomakaukau i na kēia mau waiwai: "Biperiden" "Mendileks" "biperiden hydrochloride".

"Akineton". Reviews

Ka lāʻau 'Ua nui mana i loko o ua' ōlelo ka iapaau ana o Parkinsonism tremors ma ka lala ma hope o ka pōkole manawa wā mawaena. Wahi a pono-tolerated lāʻau "Akineton".

Manaʻo Kōkua ma ka Usenet kamailio e pili ana i ka manawa kūpono o ka hoike ana mai o kekahiʻaoʻao 'ole ana e lawe i ka waiʻona.

Price "Akinetona". kahi e kuai

Ke kumu o ka pāʻoihana i ia a puni 800 rubles.

Price moʻolelo hoʻomanaʻo "Akinetona" - 560-580 rubles.

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