'O ka ma'i, Nā Hana
"Spytomin" ho'omākaukau: nā kuhikuhi no ka ho'ohana, nā hō'ailona, nā hō'ai'ē
I kēia lā e ha'i aku ana mākou i kahi ho'omākaukau me he "Spitomin". Nā kuhikuhi no ka ho'ohana'ana, ka uku, nā mana'o ho'olālā, nā analogues a me nā hi'ohi'ona - pono'ia kēia mau mea a pau i nā ma'i i kauoha'ia e kēia kauka i kēia lā'au. E'ike'oe i nā'ike kūpono a pau ma ka'atikala.
Ka wehewehe'ana o ka lā'au lā'au, kona'ano, kālepa a me ka ho'ohui'ana
He aha ka lā'au "Spitomin"? 'O nā kuhikuhi'ana no ka ho'ohana'ana ('o ka wehewehe'ana o ka lā'au lapa'au i loko o ia mea ua hō'ike'ia ma ke'ano kiko'ī) e'ōlelo ana he mau ke'oke'o kēia mau papa, he'ole, he'ōwili a he palahalaha, me kahi kiko, a me ke kūpono a me ka kahakaha'ana "E151".
'O kēia'elepa kahi'o ka busigrone hydrochloride a me nā mea kōkua like me ka carboxymethyl starch, ka lactose monohydrate, ka steium magnesium stearate, cellulosaline cellulose a me ka dioxide waipilo anhydrous.
I ke kū'ai'ana, hele mai kēia lā'au i nā pōpō a me nā pahu pahu.
Ke Kumuhana o ka hana
He aha nā'ano o ke kikowaena Spitomin? 'O nā'ōlelo a'o no ka ho'ohana (ke kumu kū'ai o nā papa i lalo iho nei)'ōlelo'ia he mea kānalua kēia no ka hui'ole benzodiazepine a he mana hana'āpana.
'A'ohe like me nā mea' ē a'eo ka no'ono'o'ole,'a'ole kēia kumu lā'au i ho'ohana'ole i nā mea hō'oki'ole, antoppilepic, sedative, hypnotic and muscle. Ke ho'okumu'ia nei kona ku'ina o ka hana ma muli o ka hopena o ka pahipirone ma nā pūnaehana dopaminerics a me nā serotonergic.
Ho'opili kēia i kēia mau lā'au i nā receptors dopamine (presynaptic) a ho'onui i ka nui o ka ho'oulu'ana o nā neurons (dopamine) o ka midbrain.
He aha nā ho'oilina'ē a'e i loko o ke kāpīpī "Spitomin"? 'O nā kuhikuhi'ana no ka ho'ohana'ana e hō'ike ana he buspirone kahi'āpana o ka'āpana o ka 5-HT1A-serotonin. 'A'ole ia e ho'opili i nā'eneke benzodiazepine a me ka GABA e pa'a,'a'ole ho'i e pili i nā hana a ka psychomotor a'a'ole e pilikia. Eia hou, 'a'ole hiki i kēia' elele ke pale i ka hana o ka mea'ona lama.
'O ka hopena maika'i o ka lā'au lapa'au i nīnau'ia e ulu mālie a mālama'ia kekahi a'elua paha ma hope o ka ho'omaka'ana o ka lā'au lapa'au.
Nā kineta o ka luna
'O ka'ae'ana o ka lā'au lapa'au "Spitomin", ke a'o'ana no ka ho'ohana'ana i kēia mea i lalo iho nei, e hana'ia ma ka'ōpala pahū. Ho'opili nui'ia'o Buspirone i ka wā e hele ai i loko o ke ake. 'O kona bioavailability he 4%, a'o ka kukuna ki'eki'e loa i ka plasma e loa'a i ka hola.
Ho'oku'u'ia'o Buspirone me ka waiū. 'O ka'ike e pili ana i ke komo'ana o kēia lā'au lapa'au i ka pale āpau ma kahi'ē.
Ke ho'opau'ia kahi lā'au lā'au me nā feces no nā hola'elima.
Hō'ike
He aha ke kumu o nā papa Spitomin? 'O ke a'o no ka ho'ohana'ana e hō'ike i nā kuhikuhi i lalo:
- Ka ma'i o ka ho'oku'u lō'ihi;
- ka iini kāna hana mea generalized;
- withdrawal maʻi pale waiʻona (me adjuvant Inc);
- panic kāna hana ;
- Nā pilikia kaumaha (e like me ke'ano o ka ancillary therapy).
Kū'ē
I loko o nā hihia hea i'ōlelo'ole'ia e ho'ohana i nā papa "Spitomin"? Ke kuhikuhi nei nā kuhikuhi no ka ho'ohana'ana i nā ma'i a me nā kūlana i ho'ohālikelike'ia ai ka lā'au:
- Glaucoma;
- Ho'oponopono i nā mea'ai o ka lā'au lapa'au;
- 'O Myasthenia gravis;
- Hō'alo i ka hō'alo'ana Renal;
- Nā makahiki makahiki;
- i ka wā hoʻokahi? eaia o Mao nā mea kūpale ;
- 'O ka manawa hana;
- 'O ka manawa o ka hāpai'ana.
Me ka lapa'au, ua kau'ia kēia māka'i no ka cirrhosis o ke ake a me ka hō'ino kīkī.
Nā lā'au lapa'au: kuhikuhi no ka ho'ohana'ana
'O nā analogs o kēia lā'au lapa'au e hō'ike'ia ma lalo nei.
Pono e lawe ka luna i ka manawa like o ka lā, ma mua a ma hope paha o ka'aina.
'A'ole pono ke ho'ohana'ia ka lā'au lapa'au (ma ke koi) e mālama i ka mana'o nui, no ka mea, kūkulu'ia ka hopena o ka lā'au ma hope o ka ho'ohana pinepine'ana.
Ho'ohana'ia nā'ano o kēia lā'au ma'amau. 'Oiai, he 15 mg. Pono e māhele'ia i 2-3 mau kau.
'O ka lā palena ho'okahi o ka lā'au lapa'au he 30 mg, a'o ka lapalapa ma'amau he 60 mg.
I ka po'e kahiko,'a'ole i koi'ia ka ho'ololi'ana o ka kau'ana. Inā hō'ino'ia nā pu'upa'a a me ka hānai, pono ke ho'ohana'ia ka lā'au me ka mālama nui a me nā kau li'ili'i.
Nā hanana pō'ino
'O ka'oihana o ka lā'au "Spitomin" kahi maika'i loa. I kekahi mau mea wale nō, e hana kēia mea hana i kekahi mau haki:
- 'O ka pehu lā'au, ka ma'i moe, ka'ele'ele, ka no'ono'o, ke kuhihewa'ana, ka headache, ka hanu'ākau;
- 'O ke kino o ke kino, ka ma'i o ka ma'i kahe, ka ho'ohemo dysphoric, ka ho'opi'i'ana o ka'ōpū o ka na'au, ka lapa'au'ana i ka ha'alū, ka'eha meocardial, dysphoria, myocardiopathy, suicidal ideation, bradycardia;
- Ka hō'ano'ana i ka pilikino, ke'ano palekana, ka euphoria, ka claustrophobia, ka hyperkinesia, ka momona, ka maka'u, ka'ili'ana i nā maka, ka mana'o'ole, nā maka'ula'ula, nā ha'alulu, ka ho'ohaunaele, ka pilikia,
- 'O ka wīwī i'ike'ia, ka laryngitis, conjunctivitis, kahe'ana o ka mucosa mīkini, nā ma'i o ka ma'i, ka kaumaha o ka umauma, nā ma'i pepeiao pepeiao, ka ma'ema'e'ole, ka'eha maka, ka'ole o ka ea, photophobia, epistaxis, ho'onui i ka pēpiko kino;
- galaktoreyu, nausea, thyroid pōʻino, flatulence, nocturnal enuresis, anorexia, ikaika loa ka makemake māhuahua, dysuria, salivation, menstrual kāna hana, intestinal kahe ana ke koko, hoolohi ejaculation a me ka 'ē aʻe.
'O ke kumu kū'ai, nā like, nā hō'ike mana'o
'O ke kumukū'ai o kēia hale he 600 mau'ūlā. Inā makemake, ua pani'ia me kahi analog like Buspiron Sandoz.
Hō'ike'ia nā mana'o mai nā mea kū'ai mai,'o ka lā'au'ona i nīnau'ia he mea hau'oli nui. Eia na'e, hiki ke lawe wale'ia no ka hana o kekahi mea lapa'au, no ka manawa lō'ihi (me ka hapalua'ole).
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